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0.0029 - 2.1
1-(beta-D-arabinofuranosyl)-cytosine
0.0003 - 1
1-(beta-D-arabinofuranosyl)-thymine
0.54 - 4.2
2',3'-dideoxycytidine
6.5
2'-deoxy-2',2'-difluorocytidine
-
0.021 - 20.6
2'-deoxyadenosine
0.00071 - 16.5
2'-deoxycytidine
0.019 - 19
2'-deoxyguanosine
0.00072 - 5.4
2'-deoxythymidine
0.817 - 1.398
2-amino-8-(1'-beta-D-2'-deoxyribofuranosyl)-imidazo[1,2-a]-1,3,5-triazin-4(8H)-one
-
0.03 - 0.037
3'-azido-2',3'-didehydro-3'-deoxythymidine
0.036 - 0.052
3'-azido-2',3'-dideoxythymidine
0.0059 - 0.4
5-(E)-(2-bromvinyl)-2'-deoxyuridine
0.00583 - 0.067
6-amino-5-nitro-3-(1'-beta-D-2'-deoxyribofuranosyl)-2(1H)-pyridone
-
0.93 - 4.2
Dideoxycytidine
additional information
additional information
-
0.0029
1-(beta-D-arabinofuranosyl)-cytosine
-
37°C, pH 7.5, wild-type enzyme
2.1
1-(beta-D-arabinofuranosyl)-cytosine
-
37°C, pH 7.5, mutant enzyme Y70W
0.0003
1-(beta-D-arabinofuranosyl)-thymine
-
37°C, pH 7.5, wild-type enzyme
1
1-(beta-D-arabinofuranosyl)-thymine
-
37°C, pH 7.5, mutant enzyme Y70W
0.54
2',3'-dideoxycytidine
-
mutant enzyme N45D/N64D
4.2
2',3'-dideoxycytidine
-
-
0.021
2'-deoxyadenosine
pH 8.0, recombinant enzyme
0.084
2'-deoxyadenosine
-
recombinant mutant A110D
0.4
2'-deoxyadenosine
-
recombinant mutant N64D
0.828
2'-deoxyadenosine
-
mutant enzyme N45D/N64D
1.1
2'-deoxyadenosine
-
recombinant mutant V84S
1.36
2'-deoxyadenosine
-
recombinant mutant V84M
1.83
2'-deoxyadenosine
-
recombinant mutant N45D
1.88
2'-deoxyadenosine
-
recombinant mutant M88R
3.2
2'-deoxyadenosine
-
recombinant mutant V84S/M88R/A110D
3.5
2'-deoxyadenosine
-
recombinant mutant V84A/M88R/A110D
3.7
2'-deoxyadenosine
-
recombinant mutant V84A
6.9
2'-deoxyadenosine
-
recombinant mutant M88R/A110D
18 - 19
2'-deoxyadenosine
-
pH 8.0, 22°C
20.6
2'-deoxyadenosine
-
recombinant wild-type enzyme
20.6
2'-deoxyadenosine
-
pH 7.8, 22°C, recombinant enzyme
20.6
2'-deoxyadenosine
pH 7.8, 22°C, recombinant enzyme
0.00071
2'-deoxycytidine
-
37°C, pH 7.5, mutant enzyme E52D
0.0012
2'-deoxycytidine
-
37°C, pH 7.5, mutant enzyme E52H
0.0162
2'-deoxycytidine
-
37°C, pH 7.5, wild-type enzyme
0.03
2'-deoxycytidine
pH 8.0, recombinant enzyme
0.055
2'-deoxycytidine
-
37°C, pH 7.5, mutant enzyme R105H
0.27
2'-deoxycytidine
-
recombinant mutant A110D
0.83
2'-deoxycytidine
-
recombinant mutant V84S
1.433
2'-deoxycytidine
wild type enzyme, at pH 7.6 and 37°C
1.6
2'-deoxycytidine
-
recombinant mutants N45D and N64D
1.62
2'-deoxycytidine
-
recombinant mutant V84S/M88R/A110D
1.8
2'-deoxycytidine
-
recombinant mutant V84M
1.94
2'-deoxycytidine
-
recombinant mutant V84A/M88R/A110D
2.1
2'-deoxycytidine
mutant enzyme Q81E, at pH 7.6 and 37°C
3.5
2'-deoxycytidine
-
recombinant mutant M88R/A110D
4.03
2'-deoxycytidine
-
mutant enzyme N45D/N64D
4.4
2'-deoxycytidine
-
recombinant mutant V84A
6.6
2'-deoxycytidine
-
37°C, pH 7.5, mutant enzyme Q81N
6.8
2'-deoxycytidine
-
37°C, pH 7.5, mutant enzyme Y70W
7.5
2'-deoxycytidine
-
recombinant mutant M88R
15
2'-deoxycytidine
-
pH 8.0, 22°C
16.5
2'-deoxycytidine
-
recombinant wild-type enzyme
16.5
2'-deoxycytidine
-
pH 7.8, 22°C, recombinant enzyme
16.5
2'-deoxycytidine
pH 7.8, 22°C, recombinant enzyme
0.019
2'-deoxyguanosine
pH 8.0, recombinant enzyme
0.073
2'-deoxyguanosine
-
recombinant mutant A110D
0.076
2'-deoxyguanosine
-
mutant enzyme N45D/N64D
0.12
2'-deoxyguanosine
-
recombinant mutant N64D
0.22
2'-deoxyguanosine
-
recombinant mutant V84M
0.64
2'-deoxyguanosine
-
recombinant mutant V84S
0.728
2'-deoxyguanosine
mutant enzyme Q81E, at pH 7.6 and 37°C
1.283
2'-deoxyguanosine
wild type enzyme, at pH 7.6 and 37°C
1.3
2'-deoxyguanosine
-
recombinant mutant N45D
1.73
2'-deoxyguanosine
-
recombinant mutant V84A/M88R/A110D
2.7
2'-deoxyguanosine
-
recombinant mutant M88R
2.8
2'-deoxyguanosine
-
recombinant mutant V84A
3.7
2'-deoxyguanosine
-
recombinant mutant M88R/A110D
4.6
2'-deoxyguanosine
-
recombinant mutant V84S/M88R/A110D
15.1
2'-deoxyguanosine
-
recombinant wild-type enzyme
15.1
2'-deoxyguanosine
-
pH 7.8, 22°C, recombinant enzyme
15.1
2'-deoxyguanosine
pH 7.8, 22°C, recombinant enzyme
18 - 19
2'-deoxyguanosine
-
pH 8.0, 22°C
0.00072
2'-deoxythymidine
-
37°C, pH 7.5, mutant enzyme E52D
0.0067
2'-deoxythymidine
-
37°C, pH 7.5, mutant enzyme R105H
0.012
2'-deoxythymidine
-
37°C, pH 7.5, mutant enzyme E52H
0.014
2'-deoxythymidine
pH 8.0, recombinant enzyme
0.0142
2'-deoxythymidine
-
37°C, pH 7.5, wild-type enzyme
0.82
2'-deoxythymidine
-
recombinant mutant N64D
2.3
2'-deoxythymidine
-
37°C, pH 7.5, mutant enzyme Y70W
2.6
2'-deoxythymidine
-
recombinant mutant N45D
5.4
2'-deoxythymidine
-
37°C, pH 7.5, mutant enzyme Q81N
0.817
2-amino-8-(1'-beta-D-2'-deoxyribofuranosyl)-imidazo[1,2-a]-1,3,5-triazin-4(8H)-one
wild type enzyme, at pH 7.6 and 37°C
-
1.398
2-amino-8-(1'-beta-D-2'-deoxyribofuranosyl)-imidazo[1,2-a]-1,3,5-triazin-4(8H)-one
mutant enzyme Q81E, at pH 7.6 and 37°C
-
0.03
3'-azido-2',3'-didehydro-3'-deoxythymidine
-
recombinant mutant N45D
0.037
3'-azido-2',3'-didehydro-3'-deoxythymidine
-
recombinant mutant N64D
0.036
3'-azido-2',3'-dideoxythymidine
-
-
0.052
3'-azido-2',3'-dideoxythymidine
-
mutant enzyme N45D/N64D
0.0059
5-(E)-(2-bromvinyl)-2'-deoxyuridine
-
37°C, pH 7.5, wild-type enzyme
0.4
5-(E)-(2-bromvinyl)-2'-deoxyuridine
-
37°C, pH 7.5, mutant enzyme Y70W
0.00583
6-amino-5-nitro-3-(1'-beta-D-2'-deoxyribofuranosyl)-2(1H)-pyridone
wild type enzyme, at pH 7.6 and 37°C
-
0.067
6-amino-5-nitro-3-(1'-beta-D-2'-deoxyribofuranosyl)-2(1H)-pyridone
mutant enzyme Q81E, at pH 7.6 and 37°C
-
0.93
Dideoxycytidine
-
recombinant mutant V84A
4.2
Dideoxycytidine
-
recombinant wild-type enzyme
0.034
thymidine
-
recombinant mutant M88R/A110D
0.037
thymidine
-
recombinant mutant V84M
0.11
thymidine
-
recombinant mutant V84A/M88R/A110D
0.13
thymidine
-
recombinant mutant M88R
0.23
thymidine
-
recombinant mutant V84S/M88R/A110D
0.35
thymidine
-
recombinant mutant A110D
0.83
thymidine
-
recombinant mutant V84S
1.22
thymidine
-
mutant enzyme N45D/N64D
2.97
thymidine
-
recombinant mutant V84A
14.2
thymidine
-
recombinant wild-type enzyme
14.2
thymidine
-
pH 7.8, 22°C, recombinant enzyme
14.2
thymidine
pH 7.8, 22°C, recombinant enzyme
15
thymidine
-
pH 8.0, 22°C
additional information
additional information
-
-
-
additional information
additional information
-
turnover-numbers of chimeric enzymes
-