Cloned (Comment) | Organism |
---|---|
expression in Escherichia coli | Giardia intestinalis |
Inhibitors | Comment | Organism | Structure |
---|---|---|---|
1,10-phenanthroline | - |
Giardia intestinalis | |
3,3'-methylene-bis(4-hydroxycoumarin) | - |
Giardia intestinalis | |
N-ethylmaleimide | - |
Giardia intestinalis | |
quercetin | - |
Giardia intestinalis | |
quinacrine dihydrochloride | 0.05 mM, 65-95% inhibition depending on substrate | Giardia intestinalis |
KM Value [mM] | KM Value Maximum [mM] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|
0.000188 | - |
menadione | cofactor NADH | Giardia intestinalis | |
0.00024 | - |
menadione | cofactor NADPH | Giardia intestinalis | |
0.000437 | - |
naphthoquinone | cofactor NADH | Giardia intestinalis | |
0.00059 | - |
naphthoquinone | cofactor NADPH | Giardia intestinalis | |
0.03 | - |
NADPH | reduction of menadione | Giardia intestinalis | |
0.033 | - |
NADPH | reduction of naphthoquinone | Giardia intestinalis | |
0.045 | - |
NADH | reduction of naphthoquinone | Giardia intestinalis | |
0.549 | - |
NADH | reduction of menadione | Giardia intestinalis |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Giardia intestinalis | - |
amitochondriate eukaryote | - |
Purification (Comment) | Organism |
---|---|
recombinant enzyme | Giardia intestinalis |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
1,4-naphthoquinone + NAD(P)H | - |
Giardia intestinalis | 1,4-naphthohydroquinone + NAD(P)+ | - |
? | |
2-methyl-1,4-naphthoquinone + NAD(P)H | - |
Giardia intestinalis | 2-methyl-1,4-naphthoquinol + NAD(P)+ | - |
? | |
3-(4,5-dimethylthiazol-2-yl)-2,5-diphenyltetrazolium bromide + NAD(P)H | - |
Giardia intestinalis | reduced 3-(4,5-dimethylthiazol-2-yl)-2,5-diphenyltetrazolium bromide + NAD(P)+ | - |
? | |
K3[Fe(CN)6] + NAD(P)H | - |
Giardia intestinalis | K4[Fe(CN)6] + NAD(P)+ | - |
? | |
menadione + NADH + H+ | - |
Giardia intestinalis | menadiol + NAD+ | - |
r | |
methyl red + NAD(P)H | - |
Giardia intestinalis | reduced methyl red + NAD(P)+ | - |
? | |
naphthoquinone + NADH + H+ | - |
Giardia intestinalis | naphthoquinol + NAD+ | - |
r |
Turnover Number Minimum [1/s] | Turnover Number Maximum [1/s] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|
23.1 | - |
menadione | cofactor NADH | Giardia intestinalis | |
29.9 | - |
naphthoquinone | cofactor NADH | Giardia intestinalis | |
31.7 | - |
NADH | reduction of menadione | Giardia intestinalis | |
34.8 | - |
menadione | cofactor NADPH | Giardia intestinalis | |
39.3 | - |
naphthoquinone | cofactor NADPH | Giardia intestinalis | |
47.5 | - |
NADPH | reduction of naphthoquinone | Giardia intestinalis | |
52.7 | - |
NADPH | reduction of menadione | Giardia intestinalis | |
62.7 | - |
NADH | reduction of naphthoquinone | Giardia intestinalis |
Ki Value [mM] | Ki Value maximum [mM] | Inhibitor | Comment | Organism | Structure |
---|---|---|---|---|---|
0.00095 | - |
dicoumarol | cofactor NADH | Giardia intestinalis | |
0.00109 | - |
dicoumarol | cofactor NADH | Giardia intestinalis | |
0.00412 | - |
dicoumarol | cofactor NADPH | Giardia intestinalis | |
0.00511 | - |
dicoumarol | cofactor NADPH | Giardia intestinalis |