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Literature summary for 2.3.1.43 extracted from

  • Nobecourt, E.; Davies, M.J.; Brown, B.E.; Curtiss, L.K.; Bonnet, D.J.; Charlton, F.; Januszewski, A.S.; Jenkins, A.J.; Barter, P.J.; Rye, K.A.
    The impact of glycation on apolipoprotein A-I structure and its ability to activate lecithin:cholesterol acyltransferase (2007), Diabetologia, 50, 643-653.
    View publication on PubMed

Activating Compound

Activating Compound Comment Organism Structure
apolipoprotein A-I glycation affects the structure of apoA-I and its ability to activate the enzyme Homo sapiens

Inhibitors

Inhibitors Comment Organism Structure
glycated discoidal (A-I)rHDL after modification of lipid-free apoA-I arginine, lysine and tryptophan residues by glucose Homo sapiens
unesterified cholesterol-(apo lipoprotein A-I-)HDL the unesterified cholesterol is deuterium-labeled Homo sapiens

Localization

Localization Comment Organism GeneOntology No. Textmining
extracellular
-
Homo sapiens
-
-

Natural Substrates/ Products (Substrates)

Natural Substrates Organism Comment (Nat. Sub.) Natural Products Comment (Nat. Pro.) Rev. Reac.
additional information Homo sapiens key enzyme in reverse cholesterol transport ?
-
?

Organism

Organism UniProt Comment Textmining
Homo sapiens
-
-
-

Purification (Commentary)

Purification (Comment) Organism
native enzyme from plasma to homogeneity Homo sapiens

Source Tissue

Source Tissue Comment Organism Textmining
plasma
-
Homo sapiens
-

Substrates and Products (Substrate)

Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
additional information key enzyme in reverse cholesterol transport Homo sapiens ?
-
?

Synonyms

Synonyms Comment Organism
LCAT
-
Homo sapiens
lecithin:cholesterol acyltransferase
-
Homo sapiens

Temperature Optimum [°C]

Temperature Optimum [°C] Temperature Optimum Maximum [°C] Comment Organism
37
-
assay at Homo sapiens

Ki Value [mM]

Ki Value [mM] Ki Value maximum [mM] Inhibitor Comment Organism Structure
additional information
-
additional information inhibition kinetics Homo sapiens