Inhibitors | Comment | Organism | Structure |
---|---|---|---|
3-(biphenyl-4-yl)-2,3-dehydroquinuclidine | 50% inhibition at 243 nM | Leishmania major | |
3-(biphenyl-4-yl)-3-hydroxyquinuclidine | 50% inhibition at 13 nM | Leishmania major | |
3-(biphenyl-4-yl)-4'[(t-butyldimethylsilyl)oxy]-3-hydroxyquinuclidine | 50% inhibition above 0.001 mM | Leishmania major | |
3-(biphenyl-4-yl-4'-hydroxy)-2,3-dehydroquinuclidine | 50% inhibition at 96 nM | Leishmania major |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Leishmania major | - |
recombinant enzyme | - |