Inhibitors | Comment | Organism | Structure |
---|---|---|---|
deoxyspergualin | - |
Homo sapiens | |
deoxyspergualin | - |
Mus musculus | |
N,N'-bis[3,5-bis[1(aminoiminomethyl)-hydrazoethyl]phenyl]decanediamide-tetrahydrochloride | i.e. CNI-1493 | Homo sapiens | |
N,N'-bis[3,5-bis[1(aminoiminomethyl)-hydrazoethyl]phenyl]decanediamide-tetrahydrochloride | i.e. CNI-1493 | Mus musculus | |
N,N'-bis[3,5-bis[1(aminoiminomethyl)-hydrazoethyl]phenyl]dodecanediamide-tetrahydrochloride | i.e. DHSI-15 | Homo sapiens | |
N,N'-bis[3,5-bis[1(aminoiminomethyl)-hydrazoethyl]phenyl]dodecanediamide-tetrahydrochloride | i.e. DHSI-15 | Mus musculus |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Homo sapiens | - |
- |
- |
Mus musculus | - |
- |
- |
Source Tissue | Comment | Organism | Textmining |
---|---|---|---|
32D cell | - |
Mus musculus | - |
BA/F3 cell | - |
Mus musculus | - |
cell culture | DHS is ubiquitously expressed in primary mouse cells and murine cell lines | Mus musculus | - |
culture condition:CD34+ cell | - |
Homo sapiens | - |
MEF cell | - |
Mus musculus | - |
additional information | DHS is ubiquitously expressed in CD34+ cellss from patients with chronic myeloid leukemia and acute myeloid leukemia | Homo sapiens | - |
NIH-3T3 cell | - |
Mus musculus | - |
NIH-3T3 cell | - |
Homo sapiens | - |
Synonyms | Comment | Organism |
---|---|---|
DHS | - |
Mus musculus |
DHS | - |
Homo sapiens |
General Information | Comment | Organism |
---|---|---|
malfunction | inhibition of proliferation of BA/F3 p210 cells including the imatinib resistant mutants M351T, E255K, and T315I by deoxyhypusine synthase inhibitors | Mus musculus |
additional information | inhibition of eIF5A by siRNA or DHS-inhibitors in combination with Imatinib exerts synergistic cytotoxic effects on BCR-ABL positive cell lines | Homo sapiens |