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Literature summary for 2.6.1.19 extracted from

  • Choi, S.Y.; Ahn, E.M.; Song, M.C.; Kim, D.W.; Kang, J.H.; Kwon, O.S.; Kang, T.C.; Baek, N.I.
    In vitro GABA-transaminase inhibitory compounds from the root of Angelica dahurica (2005), Phytother. Res., 19, 839-845.
    View publication on PubMed

Inhibitors

Inhibitors Comment Organism Structure
falcarindiol active-site directed, irreversible, 23% residual activity at 14 mM, isolate of root of Angelica dahurica Bos taurus
imperatorin active-site directed, irreversible, 14% residual activity at 14 mM, isolate of root of Angelica dahurica Bos taurus

Organism

Organism UniProt Comment Textmining
Bos taurus
-
-
-

Source Tissue

Source Tissue Comment Organism Textmining
brain
-
Bos taurus
-