Activating Compound | Comment | Organism | Structure |
---|---|---|---|
additional information | no inhibition by phosphate, the activity in higher in phosphate buffer compared to HEPES buffer | Cricetulus griseus |
Cloned (Comment) | Organism |
---|---|
expression in Escherichia coli | Cricetulus griseus |
KM Value [mM] | KM Value Maximum [mM] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|
0.0032 | - |
adenosine | recombinant enzyme, pH 7.3, 37°C, phosphate buffered saline | Cricetulus griseus | |
0.54 | - |
ribavirin | recombinant enzyme, pH 7.3, 37°C, phosphate buffered saline | Cricetulus griseus | |
7.7 | - |
viramidine | recombinant enzyme, pH 9.0, 37°C, phosphate buffered saline | Cricetulus griseus | |
7.8 | - |
ribavirin | recombinant enzyme, pH 7.3, 37°C, 0.1 M HEPES buffer | Cricetulus griseus | |
16 | - |
viramidine | recombinant enzyme, pH 7.3, 37°C, phosphate buffered saline | Cricetulus griseus |
Metals/Ions | Comment | Organism | Structure |
---|---|---|---|
Mg2+ | at 1.5 mM MgCl2 | Cricetulus griseus |
Natural Substrates | Organism | Comment (Nat. Sub.) | Natural Products | Comment (Nat. Pro.) | Rev. | Reac. |
---|---|---|---|---|---|---|
ATP + adenosine | Cricetulus griseus | - |
ADP + AMP | - |
? |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Cricetulus griseus | - |
- |
- |
Purification (Comment) | Organism |
---|---|
recombinant enzyme from Escherichia coli to homogeneity | Cricetulus griseus |
Source Tissue | Comment | Organism | Textmining |
---|---|---|---|
CHO cell | - |
Cricetulus griseus | - |
Specific Activity Minimum [µmol/min/mg] | Specific Activity Maximum [µmol/min/mg] | Comment | Organism |
---|---|---|---|
additional information | - |
- |
Cricetulus griseus |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
ATP + adenosine | - |
Cricetulus griseus | ADP + AMP | - |
? | |
ATP + ribavirin | very low activity | Cricetulus griseus | ADP + ribavirin 5'-phosphate | - |
? | |
ATP + viramidine | very low activity | Cricetulus griseus | ADP + viramidine 5'-phosphate | - |
? |
Temperature Optimum [°C] | Temperature Optimum Maximum [°C] | Comment | Organism |
---|---|---|---|
37 | - |
assay at | Cricetulus griseus |
Turnover Number Minimum [1/s] | Turnover Number Maximum [1/s] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|
0.16 | - |
viramidine | recombinant enzyme, pH 7.3, 37°C, phosphate buffered saline | Cricetulus griseus | |
0.26 | - |
viramidine | recombinant enzyme, pH 9.0, 37°C, phosphate buffered saline | Cricetulus griseus | |
0.62 | - |
ribavirin | recombinant enzyme, pH 7.3, 37°C, 0.1 M HEPES buffer | Cricetulus griseus | |
1.8 | - |
ribavirin | recombinant enzyme, pH 7.3, 37°C, phosphate buffered saline | Cricetulus griseus | |
13 | - |
adenosine | recombinant enzyme, pH 7.3, 37°C, phosphate buffered saline | Cricetulus griseus |
pH Optimum Minimum | pH Optimum Maximum | Comment | Organism |
---|---|---|---|
7.3 | - |
assay at | Cricetulus griseus |