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Literature summary for 2.7.1.21 extracted from

  • Chello, P.L.; Jaffe, J.J.
    Comparative properties of trypanosomal and mammalian thymidine kinases (1972), Comp. Biochem. Physiol. B, 43, 543-562.
    View publication on PubMed

Inhibitors

Inhibitors Comment Organism Structure
dTTP
-
Rattus norvegicus
dTTP
-
Trypanosoma brucei rhodesiense
suramin
-
Rattus norvegicus
suramin
-
Trypanosoma brucei rhodesiense

KM Value [mM]

KM Value [mM] KM Value Maximum [mM] Substrate Comment Organism Structure
additional information
-
additional information
-
Rattus norvegicus
additional information
-
additional information
-
Trypanosoma brucei rhodesiense

Metals/Ions

Metals/Ions Comment Organism Structure
Ca2+ not Rattus norvegicus
Ca2+ not Trypanosoma brucei rhodesiense
Co2+ can partially substitute for Mg2+ Rattus norvegicus
Co2+ can partially substitute for Mg2+ Trypanosoma brucei rhodesiense
Mg2+
-
Rattus norvegicus
Mg2+
-
Trypanosoma brucei rhodesiense
additional information inactive with Ba2+ and Ca2+ Rattus norvegicus
additional information inactive with Ba2+ and Ca2+ Trypanosoma brucei rhodesiense
Zn2+ liver Rattus norvegicus

Organism

Organism UniProt Comment Textmining
Rattus norvegicus
-
-
-
Trypanosoma brucei rhodesiense
-
blood stream and epimastigote form
-

Source Tissue

Source Tissue Comment Organism Textmining
epimastigote
-
Trypanosoma brucei rhodesiense
-
liver
-
Rattus norvegicus
-

Substrates and Products (Substrate)

Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
additional information comparison rat liver, Trypanosoma brucei Rattus norvegicus ?
-
?
additional information comparison rat liver, Trypanosoma brucei Trypanosoma brucei rhodesiense ?
-
?