Activating Compound | Comment | Organism | Structure |
---|---|---|---|
histone | stimulates | Homo sapiens | |
phosvitin | stimulates | Homo sapiens | |
poly(L-lysine) | stimulates | Homo sapiens | |
Polyarginine | stimulates | Homo sapiens | |
spermidine | half-maximal stimulation at 1.5 mM | Homo sapiens |
Inhibitors | Comment | Organism | Structure |
---|---|---|---|
2'-dATP | - |
Homo sapiens | |
3'-dATP | - |
Homo sapiens | |
8-bromo-ATP | - |
Homo sapiens | |
adenosine | - |
Homo sapiens | |
ADP | - |
Homo sapiens | |
AMP | - |
Homo sapiens | |
cAMP | - |
Homo sapiens | |
GTP | - |
Homo sapiens | |
N6-dimethylamine-adenosine 5'-triphosphate | - |
Homo sapiens |
KM Value [mM] | KM Value Maximum [mM] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|
0.02 | - |
ATP | pH 7.4, 25°C | Homo sapiens |
Localization | Comment | Organism | GeneOntology No. | Textmining |
---|---|---|---|---|
membrane | - |
Homo sapiens | 16020 | - |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Homo sapiens | - |
- |
- |
Source Tissue | Comment | Organism | Textmining |
---|---|---|---|
A-431 cell | - |
Homo sapiens | - |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
ATP + 1-phosphatidyl-1D-myo-inositol | - |
Homo sapiens | ADP + 1-phosphatidyl-1D-myo-inositol 4-phosphate | - |
? |
Ki Value [mM] | Ki Value maximum [mM] | Inhibitor | Comment | Organism | Structure |
---|---|---|---|---|---|
0.01 | - |
ADP | pH 7.4, 25°C, in absence of spermidine | Homo sapiens | |
0.012 | - |
3'-dATP | pH 7.4, 25°C, in absence of spermidine | Homo sapiens | |
0.013 | - |
GTP | pH 7.4, 25°C, in absence of spermidine | Homo sapiens | |
0.014 | - |
2'-dATP | pH 7.4, 25°C, in presence of 3 mM spermidine | Homo sapiens | |
0.04 | - |
N6-dimethylamine-adenosine 5'-triphosphate | pH 7.4, 25°C, in presence of 3 mM spermidine | Homo sapiens | |
0.07 | - |
adenosine | pH 7.4, 25°C, in absence of spermidine | Homo sapiens | |
0.11 | - |
8-bromo-ATP | pH 7.4, 25°C, in presence of 3 mM spermidine | Homo sapiens | |
0.5 | - |
cAMP | pH 7.4, 25°C, in absence of spermidine | Homo sapiens | |
0.53 | - |
AMP | pH 7.4, 25°C, in absence of spermidine | Homo sapiens | |
1.9 | - |
N6-dimethylamine-adenosine 5'-triphosphate | pH 7.4, 25°C, in absence of spermidine | Homo sapiens |