Cloned (Comment) | Organism |
---|---|
expression in Escherichia coli strain M15 | Plasmodium falciparum |
Inhibitors | Comment | Organism | Structure |
---|---|---|---|
additional information | not inhibitory: atractyloside, chloroquine, primaquine, artemisinine, mefloquine | Plasmodium falciparum | |
P1,P5-di(adenosine-5')pentaphosphate | - |
Plasmodium falciparum |
KM Value [mM] | KM Value Maximum [mM] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|
0.05 | - |
AMP | pH 6.0 and pH 7.4 | Plasmodium falciparum | |
0.12 | - |
ATP | pH 7.4 | Plasmodium falciparum | |
0.13 | - |
ATP | pH 6.0 | Plasmodium falciparum |
Molecular Weight [Da] | Molecular Weight Maximum [Da] | Comment | Organism |
---|---|---|---|
27600 | - |
calculated without His-tag | Plasmodium falciparum |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Plasmodium falciparum | Q7Z0H0 | strains HB3 and Dd2 | - |
Purification (Comment) | Organism |
---|---|
- |
Plasmodium falciparum |
Specific Activity Minimum [µmol/min/mg] | Specific Activity Maximum [µmol/min/mg] | Comment | Organism |
---|---|---|---|
additional information | - |
Vmax 75 1 mM at pH 6.0 and 25°C | Plasmodium falciparum |
100 | - |
wild type AK | Plasmodium falciparum |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
ATP + AMP | - |
Plasmodium falciparum | ADP + ADP | - |
? | |
CTP + AMP | - |
Plasmodium falciparum | CDP + ADP | - |
? | |
GTP + AMP | - |
Plasmodium falciparum | GDP + ADP | - |
? | |
ITP + AMP | - |
Plasmodium falciparum | IDP + ADP | - |
? | |
additional information | monophosphates: IMP, GMP, CMP, UMP: activity below 1% | Plasmodium falciparum | ? | - |
? | |
UTP + AMP | - |
Plasmodium falciparum | UDP + ADP | - |
? |
Ki Value [mM] | Ki Value maximum [mM] | Inhibitor | Comment | Organism | Structure |
---|---|---|---|---|---|
0.0001 | - |
P1,P5-di(adenosine-5')pentaphosphate | pH 7.4 | Plasmodium falciparum | |
0.00038 | - |
P1,P5-di(adenosine-5')pentaphosphate | pH 6 | Plasmodium falciparum |