Cloned (Comment) | Organism |
---|---|
expressed in Escherichia coli BL21 cells | Human immunodeficiency virus 1 |
Crystallization (Comment) | Organism |
---|---|
in complex with inhibitor TMC278, hanging drop vapour diffusion method, using 9% to 12% PEG 8000, 50 mM imidazole pH 6.0-6.8, 10 mM spermine, 15 mM MgSO4 and 100 mM ammonium sulfate | Human immunodeficiency virus 1 |
Inhibitors | Comment | Organism | Structure |
---|---|---|---|
Etravirine | - |
Human immunodeficiency virus 1 | |
Rilpivirine | - |
Human immunodeficiency virus 1 | |
TMC125 | - |
Human immunodeficiency virus 1 | |
TMC278 | nonnucleoside reverse transcriptase inhibitor | Human immunodeficiency virus 1 |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Human immunodeficiency virus 1 | P03366 | - |
- |
Purification (Comment) | Organism |
---|---|
Mono Q column chromatography | Human immunodeficiency virus 1 |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
deoxynucleoside triphosphate + DNAn | - |
Human immunodeficiency virus 1 | diphosphate + DNAn+1 | - |
? |
Synonyms | Comment | Organism |
---|---|---|
reverse transcriptase | - |
Human immunodeficiency virus 1 |