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Literature summary for 1.10.3.9 extracted from

  • Jampilek, J.; Kralova, K.; Pesko, M.; Kos, J.
    Ring-substituted 8-hydroxyquinoline-2-carboxanilides as photosystem II inhibitors (2016), Bioorg. Med. Chem. Lett., 26, 3862-3865 .
    View publication on PubMed
Search for more literature for 1.10.3.9

Inhibitors

Inhibitors Comment Organism Structure
3-(3,4-dichlorophenyl)-1,1-dimethylurea
-
 Spinacia oleracea
8-hydroxy-N-(3-methylphenyl)quinoline-2-carboxamide
-
 Spinacia oleracea
additional information inhibitory efficiency of ring-substituted 8-hydroxyquinoline-2-carboxanilides depends on the compound lipophilicity, the electronic properties of the substituent R and the position of the substituent R on the benzene ring. Compounds probably bind the section between P680 and plastoquinone QB on the acceptor side of PS II Spinacia oleracea
N-(3-fluorophenyl)-8-hydroxyquinoline-2-carboxamide
-
 Spinacia oleracea

Localization

Localization Comment Organism GeneOntology No. Textmining
chloroplast
-
 Spinacia oleracea 9507
-

Organism

Organism UniProt Comment Textmining
Spinacia oleracea
-
-
-

Substrates and Products (Substrate)

Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
H2O + 2,6-dichlorophenolindophenol + hv
-
 Spinacia oleracea O2 + reduced 2,6-dichlorophenolindophenol
-
 ?

IC50 Value

IC50 Value IC50 Value Maximum Comment Organism Inhibitor Structure
0.0019
-
 pH not specified in the publication, temperature not specified in the publication Spinacia oleracea 3-(3,4-dichlorophenyl)-1,1-dimethylurea
0.0023
-
 pH not specified in the publication, temperature not specified in the publication Spinacia oleracea N-(3-fluorophenyl)-8-hydroxyquinoline-2-carboxamide
0.0027
-
 pH not specified in the publication, temperature not specified in the publication Spinacia oleracea 8-hydroxy-N-(3-methylphenyl)quinoline-2-carboxamide