Inhibitors | Comment | Organism | Structure |
---|---|---|---|
3,5-diamino-1H-1,2,4-triazole | 2.3 mM, 50% inhibition of CDP reduction, 2.6 mM, 50% inhibition of ADP reduction | Mesocricetus auratus | |
ADP | - |
Mesocricetus auratus | |
ATP | CDP reduction is inhibited by free ATP | Mesocricetus auratus | |
CDP | - |
Mesocricetus auratus | |
dADP | product inhibition | Mesocricetus auratus | |
dATP | 2.1 mM, 50% inhibition; inhibition of CDP reduction; weak inhibition of ADP reduction | Mesocricetus auratus | |
dCDP | product inhibition | Mesocricetus auratus | |
dCTP | 1.2 mM, 50% inhibition of CDP reduction, 0.89 mM, 50% inhibition of ADP reduction | Mesocricetus auratus | |
dGDP | product inhibition | Mesocricetus auratus | |
dGTP | 1.2 mM, 50% inhibition of CDP reduction, 0.93 mM, 50% inhibition of ADP reduction | Mesocricetus auratus | |
dTTP | inhibition of CDP reduction | Mesocricetus auratus | |
dUDP | product inhibition | Mesocricetus auratus | |
EDTA | - |
Mesocricetus auratus | |
GDP | - |
Mesocricetus auratus | |
Hydroxyurea | - |
Mesocricetus auratus | |
Mg2+ | uncomplexed Mg2+ | Mesocricetus auratus | |
additional information | each ribonucleoside diphosphate substrate is competitively inhibited by reduction of each other substrate | Mesocricetus auratus | |
UDP | - |
Mesocricetus auratus |
KM Value [mM] | KM Value Maximum [mM] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|
0.00065 | - |
CDP | - |
Mesocricetus auratus | |
0.0012 | - |
GDP | - |
Mesocricetus auratus | |
0.012 | - |
ADP | - |
Mesocricetus auratus | |
0.08 | - |
UDP | - |
Mesocricetus auratus |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Mesocricetus auratus | - |
baby hamster kidney cells, enzyme induced by Herpes simplex, virus type 1, HSV-1 | - |
Source Tissue | Comment | Organism | Textmining |
---|---|---|---|
BHK-21 cell | - |
Mesocricetus auratus | - |
kidney | baby hamster kidney cells | Mesocricetus auratus | - |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
ADP + thioredoxin | - |
Mesocricetus auratus | 2'-dADP + thioredoxin disulfide + H2O | - |
r | |
CDP + thioredoxin | - |
Mesocricetus auratus | 2'-dCDP + thioredoxin disulfide + H2O | - |
r | |
GDP + thioredoxin | - |
Mesocricetus auratus | 2'-dGDP + thioredoxin disulfide + H2O | - |
r | |
ribonucleoside diphosphate + reduced thioredoxin | - |
Mesocricetus auratus | 2'-deoxyribonucleoside diphosphate + oxidized thioredoxin + H2O | - |
ir | |
UDP + reduced thioredoxin | - |
Mesocricetus auratus | 2'-deoxy-UDP + oxidized thioredoxin + H2O | - |
? |
pH Optimum Minimum | pH Optimum Maximum | Comment | Organism |
---|---|---|---|
8.1 | - |
- |
Mesocricetus auratus |
Ki Value [mM] | Ki Value maximum [mM] | Inhibitor | Comment | Organism | Structure |
---|---|---|---|---|---|
0.00058 | - |
CDP | vs. GDP | Mesocricetus auratus | |
0.0006 | - |
GDP | vs. ADP | Mesocricetus auratus | |
0.0007 | - |
CDP | vs. ADP | Mesocricetus auratus | |
0.0012 | - |
GDP | vs. CDP | Mesocricetus auratus | |
0.0018 | - |
GDP | vs. UDP | Mesocricetus auratus | |
0.0019 | - |
CDP | vs. UDP | Mesocricetus auratus | |
0.0055 | - |
ADP | vs. GDP | Mesocricetus auratus | |
0.0058 | - |
UDP | vs. GDP | Mesocricetus auratus | |
0.014 | - |
ADP | vs. CDP | Mesocricetus auratus | |
0.036 | - |
ADP | vs. UDP | Mesocricetus auratus | |
0.042 | - |
UDP | vs. CDP | Mesocricetus auratus | |
0.043 | - |
UDP | vs. ADP | Mesocricetus auratus |