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Literature summary for 1.8.4.2 extracted from

  • Roth, R.A.
    Bacitracin: an inhibitor of the insulin degrading activity of glutathione-insulin transhydrogenase (1981), Biochem. Biophys. Res. Commun., 98, 431-438.
    View publication on PubMed

Inhibitors

Inhibitors Comment Organism Structure
bacitracin antibiotic Rattus norvegicus

KM Value [mM]

KM Value [mM] KM Value Maximum [mM] Substrate Comment Organism Structure
0.004
-
Insulin
-
Rattus norvegicus

Natural Substrates/ Products (Substrates)

Natural Substrates Organism Comment (Nat. Sub.) Natural Products Comment (Nat. Pro.) Rev. Reac.
GSH + protein disulfide Rattus norvegicus
-
GSSG + protein-dithiol
-
?

Organism

Organism UniProt Comment Textmining
Rattus norvegicus
-
-
-

Purification (Commentary)

Purification (Comment) Organism
-
Rattus norvegicus

Source Tissue

Source Tissue Comment Organism Textmining
liver
-
Rattus norvegicus
-

Specific Activity [micromol/min/mg]

Specific Activity Minimum [µmol/min/mg] Specific Activity Maximum [µmol/min/mg] Comment Organism
additional information
-
-
Rattus norvegicus

Substrates and Products (Substrate)

Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
GSH + protein disulfide
-
Rattus norvegicus GSSG + protein-dithiol
-
?