Inhibitors | Comment | Organism | Structure |
---|---|---|---|
2-Bromolysergic acid diethylamide | - |
Cavia porcellus | |
bromo-lysergic acid diethylamide | 55% inhibition at 0.005 mM | Cavia porcellus | |
Bufotenine | - |
Cavia porcellus | |
chlorpromazine | 60% inhibition at o.oo5 mM | Cavia porcellus | |
chlorpromazine | - |
Felis catus | |
chlorpromazine | - |
Mus musculus | |
chlorpromazine | - |
Oryctolagus cuniculus | |
chlorpromazine | - |
Rattus norvegicus | |
Methylhistamine | 40% inhibition at 0.1 mM | Cavia porcellus | |
Methylhistamine | - |
Rattus norvegicus | |
p-chloromercuribenzoate | 90% inhibition at 0.01 mM | Cavia porcellus | |
p-chloromercuribenzoate | - |
Rattus norvegicus | |
serotonin | 33% inhibition at 0.005 mM | Cavia porcellus | |
serotonin | - |
Felis catus | |
serotonin | - |
Mus musculus | |
serotonin | - |
Oryctolagus cuniculus | |
serotonin | - |
Rattus norvegicus | |
Tubocurare | - |
Cavia porcellus |
KM Value [mM] | KM Value Maximum [mM] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|
0.035 | - |
histamine | - |
Cavia porcellus | |
0.38 | - |
S-adenosyl-L-methionine | - |
Cavia porcellus |
Localization | Comment | Organism | GeneOntology No. | Textmining |
---|---|---|---|---|
soluble | - |
Cavia porcellus | - |
- |
soluble | - |
Mus musculus | - |
- |
soluble | - |
Rattus norvegicus | - |
- |
soluble | - |
Oryctolagus cuniculus | - |
- |
soluble | - |
Felis catus | - |
- |
Natural Substrates | Organism | Comment (Nat. Sub.) | Natural Products | Comment (Nat. Pro.) | Rev. | Reac. |
---|---|---|---|---|---|---|
additional information | Cavia porcellus | major pathway of histamine metabolism in mammals | ? | - |
? | |
additional information | Mus musculus | major pathway of histamine metabolism in mammals | ? | - |
? | |
additional information | Rattus norvegicus | major pathway of histamine metabolism in mammals | ? | - |
? | |
additional information | Oryctolagus cuniculus | major pathway of histamine metabolism in mammals | ? | - |
? | |
additional information | Felis catus | major pathway of histamine metabolism in mammals | ? | - |
? |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Cavia porcellus | - |
- |
- |
Felis catus | - |
- |
- |
Mus musculus | - |
- |
- |
Oryctolagus cuniculus | - |
- |
- |
Rattus norvegicus | - |
- |
- |
Purification (Comment) | Organism |
---|---|
- |
Cavia porcellus |
Source Tissue | Comment | Organism | Textmining |
---|---|---|---|
abdomen | abdominal skin | Cavia porcellus | - |
abdomen | abdominal skin | Mus musculus | - |
abdomen | abdominal skin | Rattus norvegicus | - |
abdomen | abdominal skin | Oryctolagus cuniculus | - |
abdomen | abdominal skin | Felis catus | - |
adrenal gland | - |
Cavia porcellus | - |
adrenal gland | - |
Oryctolagus cuniculus | - |
adrenal gland | - |
Felis catus | - |
brain | - |
Cavia porcellus | - |
brain | - |
Mus musculus | - |
brain | - |
Rattus norvegicus | - |
brain | - |
Oryctolagus cuniculus | - |
brain | - |
Felis catus | - |
heart | - |
Cavia porcellus | - |
heart | - |
Mus musculus | - |
heart | - |
Rattus norvegicus | - |
heart | - |
Oryctolagus cuniculus | - |
heart | - |
Felis catus | - |
ileum | - |
Cavia porcellus | - |
ileum | - |
Rattus norvegicus | - |
ileum | - |
Oryctolagus cuniculus | - |
ileum | - |
Felis catus | - |
kidney | - |
Cavia porcellus | - |
kidney | - |
Mus musculus | - |
kidney | - |
Rattus norvegicus | - |
kidney | - |
Oryctolagus cuniculus | - |
kidney | - |
Felis catus | - |
liver | - |
Cavia porcellus | - |
liver | - |
Mus musculus | - |
liver | - |
Oryctolagus cuniculus | - |
liver | - |
Felis catus | - |
liver | not in rat | Rattus norvegicus | - |
lung | - |
Cavia porcellus | - |
lung | - |
Mus musculus | - |
lung | - |
Oryctolagus cuniculus | - |
lung | - |
Felis catus | - |
lung | not in rat | Rattus norvegicus | - |
pancreas | - |
Felis catus | - |
sciatic nerve | - |
Cavia porcellus | - |
sciatic nerve | - |
Oryctolagus cuniculus | - |
sciatic nerve | - |
Felis catus | - |
spleen | - |
Cavia porcellus | - |
spleen | - |
Mus musculus | - |
spleen | - |
Oryctolagus cuniculus | - |
spleen | - |
Felis catus | - |
spleen | not in rat | Rattus norvegicus | - |
stomach | - |
Cavia porcellus | - |
stomach | - |
Mus musculus | - |
stomach | - |
Oryctolagus cuniculus | - |
stomach | - |
Felis catus | - |
thigh muscle | - |
Cavia porcellus | - |
thigh muscle | - |
Mus musculus | - |
thigh muscle | - |
Rattus norvegicus | - |
thigh muscle | - |
Oryctolagus cuniculus | - |
thigh muscle | - |
Felis catus | - |
trachea | - |
Cavia porcellus | - |
trachea | - |
Felis catus | - |
Specific Activity Minimum [µmol/min/mg] | Specific Activity Maximum [µmol/min/mg] | Comment | Organism |
---|---|---|---|
25.4 | - |
- |
Cavia porcellus |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
additional information | major pathway of histamine metabolism in mammals | Cavia porcellus | ? | - |
? | |
additional information | major pathway of histamine metabolism in mammals | Mus musculus | ? | - |
? | |
additional information | major pathway of histamine metabolism in mammals | Rattus norvegicus | ? | - |
? | |
additional information | major pathway of histamine metabolism in mammals | Oryctolagus cuniculus | ? | - |
? | |
additional information | major pathway of histamine metabolism in mammals | Felis catus | ? | - |
? | |
S-adenosyl-L-methionine + histamine | - |
Cavia porcellus | S-adenosyl-L-homocysteine + Ntau-methylhistamine | - |
? | |
S-adenosyl-L-methionine + histamine | - |
Mus musculus | S-adenosyl-L-homocysteine + Ntau-methylhistamine | - |
? | |
S-adenosyl-L-methionine + histamine | - |
Rattus norvegicus | S-adenosyl-L-homocysteine + Ntau-methylhistamine | - |
? | |
S-adenosyl-L-methionine + histamine | - |
Oryctolagus cuniculus | S-adenosyl-L-homocysteine + Ntau-methylhistamine | - |
? | |
S-adenosyl-L-methionine + histamine | - |
Felis catus | S-adenosyl-L-homocysteine + Ntau-methylhistamine | - |
? |
Temperature Optimum [°C] | Temperature Optimum Maximum [°C] | Comment | Organism |
---|---|---|---|
37 | - |
assay at | Cavia porcellus |
37 | - |
assay at | Mus musculus |
37 | - |
assay at | Rattus norvegicus |
37 | - |
assay at | Oryctolagus cuniculus |
37 | - |
assay at | Felis catus |
pH Optimum Minimum | pH Optimum Maximum | Comment | Organism |
---|---|---|---|
7.2 | 7.4 | - |
Cavia porcellus |
7.2 | 7.4 | - |
Mus musculus |