Inhibitors | Comment | Organism | Structure |
---|---|---|---|
5'-GMP | reversible and uncompetitive inhibition | Leishmania amazonensis | |
beta,gamma-methylene-GTP | - |
Leishmania amazonensis | |
GDP | - |
Leishmania amazonensis | |
GTP | - |
Leishmania amazonensis | |
guanosine | - |
Leishmania amazonensis | |
guanosine tetraphosphate | - |
Leishmania amazonensis |
KM Value [mM] | KM Value Maximum [mM] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|
0.0002 | - |
3'-AMP | at pH 7.4 and 25°C | Leishmania amazonensis |
Natural Substrates | Organism | Comment (Nat. Sub.) | Natural Products | Comment (Nat. Pro.) | Rev. | Reac. |
---|---|---|---|---|---|---|
a 3'-ribonucleotide + H2O | Leishmania amazonensis | - |
a ribonucleoside + phosphate | - |
? | |
a 3'-ribonucleotide + H2O | Leishmania amazonensis MHOM/BR/75/Josefa | - |
a ribonucleoside + phosphate | - |
? |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Leishmania amazonensis | - |
- |
- |
Leishmania amazonensis MHOM/BR/75/Josefa | - |
- |
- |
Source Tissue | Comment | Organism | Textmining |
---|---|---|---|
promastigote | - |
Leishmania amazonensis | - |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
3'-AMP + H2O | - |
Leishmania amazonensis | adenosine + phosphate | - |
? | |
3'-AMP + H2O | - |
Leishmania amazonensis MHOM/BR/75/Josefa | adenosine + phosphate | - |
? | |
a 3'-ribonucleotide + H2O | - |
Leishmania amazonensis | a ribonucleoside + phosphate | - |
? | |
a 3'-ribonucleotide + H2O | - |
Leishmania amazonensis MHOM/BR/75/Josefa | a ribonucleoside + phosphate | - |
? |
Synonyms | Comment | Organism |
---|---|---|
3'-NT | - |
Leishmania amazonensis |
3'-NT/Nu | - |
Leishmania amazonensis |
ecto-3'-nucleotidase | - |
Leishmania amazonensis |
ecto-3'-nucleotidase/nuclease | - |
Leishmania amazonensis |
Ki Value [mM] | Ki Value maximum [mM] | Inhibitor | Comment | Organism | Structure |
---|---|---|---|---|---|
0.00371 | - |
GDP | at pH 7.4 and 25°C | Leishmania amazonensis | |
0.00479 | - |
5'-GMP | at pH 7.4 and 25°C | Leishmania amazonensis | |
0.00503 | - |
GTP | at pH 7.4 and 25°C | Leishmania amazonensis | |
0.01732 | - |
beta,gamma-methylene-GTP | at pH 7.4 and 25°C | Leishmania amazonensis | |
0.03229 | - |
guanosine | at pH 7.4 and 25°C | Leishmania amazonensis | |
0.05663 | - |
guanosine tetraphosphate | at pH 7.4 and 25°C | Leishmania amazonensis |