Activating Compound | Comment | Organism | Structure |
---|---|---|---|
dithiothreitol | presence of disulfide-reducing agent such as dithiothreitol required | Bos taurus |
Inhibitors | Comment | Organism | Structure |
---|---|---|---|
1,10-phenanthroline | - |
Bos taurus | |
2-Iodoacetamide | - |
Bos taurus | |
2-Pyrrolidone | - |
Bos taurus | |
Cd2+ | - |
Bos taurus | |
Cu2+ | - |
Bos taurus | |
Hg2+ | - |
Bos taurus | |
NEM | - |
Bos taurus | |
p-hydroxymercuribenzoate | - |
Bos taurus | |
Zn2+ | - |
Bos taurus |
KM Value [mM] | KM Value Maximum [mM] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|
0.01364 | - |
pyroglutamyl-His-Pro-4-methylcoumarin 7-amide | - |
Bos taurus | |
0.01536 | - |
pyroglutamyl-4-methylcoumarin 7-amide | - |
Bos taurus | |
0.02076 | - |
Pyroglutamyl-beta-naphthylamide | - |
Bos taurus |
Molecular Weight [Da] | Molecular Weight Maximum [Da] | Comment | Organism |
---|---|---|---|
23700 | - |
gel filtration | Bos taurus |
24000 | - |
1 * 24000, SDS-PAGE | Bos taurus |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Bos taurus | - |
- |
- |
Purification (Comment) | Organism |
---|---|
- |
Bos taurus |
Source Tissue | Comment | Organism | Textmining |
---|---|---|---|
brain | - |
Bos taurus | - |
Specific Activity Minimum [µmol/min/mg] | Specific Activity Maximum [µmol/min/mg] | Comment | Organism |
---|---|---|---|
additional information | - |
- |
Bos taurus |
Storage Stability | Organism |
---|---|
-80°C, 17% loss of activity after 4 weeks | Bos taurus |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
bombesin + H2O | - |
Bos taurus | pyroglutamate + Gln-Arg-Leu-Gly-Asn-Gln-Trp-Ala-Val-Gly-His-Leu-Met-NH2 | - |
? | |
L-pyroglutamyl-His-Pro-4-methylcoumarin 7-amide + H2O | - |
Bos taurus | L-pyroglutamate + His-Pro-4-methylcoumarin 7-amide | - |
? | |
luteinizing-hormone-releasing hormone + H2O | - |
Bos taurus | ? | - |
? | |
neurotensin + H2O | - |
Bos taurus | pyroglutamate + Leu-Tyr-Glu-Asn-Lys-Pro-Ag-Arg-Pro-Tyr-Ile-Leu | - |
? | |
pyroglutamyl-4-methylcoumarin 7-amide + H2O | - |
Bos taurus | pyroglutamate + 7-amino-4-methylcoumarin | - |
? | |
pyroglutamyl-beta-naphthylamide + H2O | - |
Bos taurus | pyroglutamate + beta-naphthylamine | - |
? | |
thyroliberin + H2O | - |
Bos taurus | pyroglutamate + His-Pro-NH2 | - |
? |
Subunits | Comment | Organism |
---|---|---|
monomer | 1 * 24000, SDS-PAGE | Bos taurus |
pH Optimum Minimum | pH Optimum Maximum | Comment | Organism |
---|---|---|---|
8.5 | - |
- |
Bos taurus |