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Literature summary for 3.4.21.39 extracted from

  • Kido, H.; Fukusen, N.; Katunuma, N.
    Chymotrypsin- and trypsin-type serine proteases in rat mast cells: properties and functions (1985), Arch. Biochem. Biophys., 239, 436-443.
    View publication on PubMed

Inhibitors

Inhibitors Comment Organism Structure
alpha1-Aantichymotrypsin
-
Rattus norvegicus
alpha1-antitrypsin
-
Rattus norvegicus
antipain
-
Rattus norvegicus
Aprotinin
-
Rattus norvegicus
bestatin
-
Rattus norvegicus
decanoyl lysophosphatidic acid
-
Rattus norvegicus
diisopropyl fluorophosphate
-
Rattus norvegicus
dilauroyl phosphatidic acid
-
Rattus norvegicus
dioleoyl phosphatidic acid
-
Rattus norvegicus
dipalmitoyl phosphatidic acid
-
Rattus norvegicus
distearoyl phosphatidic acid
-
Rattus norvegicus
elaidic acid
-
Rattus norvegicus
linoleic acid
-
Rattus norvegicus
linolenic acid
-
Rattus norvegicus
oleamide
-
Rattus norvegicus
oleic acid
-
Rattus norvegicus
oleoyl lysophosphatidic acid
-
Rattus norvegicus
palmitoyl lysophosphatidic acid
-
Rattus norvegicus
phosphatidic acid from bovine brain Rattus norvegicus
phosphatidylethanolamine
-
Rattus norvegicus
phosphatidylinositol
-
Rattus norvegicus
phosphatidylserine
-
Rattus norvegicus
Soybean trypsin inhibitor
-
Rattus norvegicus
stearic acid
-
Rattus norvegicus

Natural Substrates/ Products (Substrates)

Natural Substrates Organism Comment (Nat. Sub.) Natural Products Comment (Nat. Pro.) Rev. Reac.
additional information Rattus norvegicus the enzyme plays a crucial or significant role in the process of degranulation ?
-
?

Organism

Organism UniProt Comment Textmining
Rattus norvegicus
-
-
-

Purification (Commentary)

Purification (Comment) Organism
-
Rattus norvegicus

Source Tissue

Source Tissue Comment Organism Textmining
mast cell
-
Rattus norvegicus
-
peritoneum
-
Rattus norvegicus
-

Substrates and Products (Substrate)

Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
benzoyl-Arg-4-methylcoumarin 7-amide + H2O 1.2% of the activity with succinyl-Leu-Leu-Val-Tyr-4-methylcoumarin 7-amide Rattus norvegicus benzoyl-Arg + 4-methylcoumarin 7-amide
-
?
additional information the enzyme plays a crucial or significant role in the process of degranulation Rattus norvegicus ?
-
?
Pro-Phe-Arg-4-methylcoumarin 7-amide + H2O 4.6% of the activity with succinyl-Leu-Leu-Val-Tyr-4-methylcoumarin 7-amide Rattus norvegicus ?
-
?
Succinyl-Ala-Ala-Pro-Phe-4-methylcoumarin 7-amide + H2O 26.6% of the activity with succinyl-Leu-Leu-Val-Tyr-4-methylcoumarin 7-amide Rattus norvegicus ?
-
?
succinyl-Leu-Leu-Val-Tyr-4-methylcoumarin 7-amide + H2O
-
Rattus norvegicus ?
-
?
t-butyloxycarbonyl-Val-Leu-Lys-4-methylcoumarin 7-amide + H2O 2.6% of the activity with succinyl-Leu-Leu-Val-Tyr-4-methylcoumarin 7-amide Rattus norvegicus ?
-
?