Activating Compound | Comment | Organism | Structure |
---|---|---|---|
2-mercaptoethanol | activates | Homo sapiens | |
cysteine | activates | Homo sapiens | |
dithiothreitol | activates | Homo sapiens |
Inhibitors | Comment | Organism | Structure |
---|---|---|---|
iodoacetic acid | - |
Homo sapiens | |
L-3-carboxy-2,3-trans-epoxypropionyl-leucylamido-(4-guanidino)butane | E-64 | Homo sapiens | |
leupeptin | - |
Homo sapiens |
KM Value [mM] | KM Value Maximum [mM] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|
0.012 | - |
benzyloxycarbonyl-Val-Lys-Lys-Arg-4-methoxy-beta-naphthylamide | - |
Homo sapiens | |
0.022 | - |
benzyloxycarbonyl-Ala-Arg-Arg-4-methoxy-beta-naphthylamide | - |
Homo sapiens | |
0.038 | - |
benzyloxycarbonyl-Arg-Arg-4-methylcoumaryl-7-amide | - |
Homo sapiens | |
0.038 | - |
benzyloxycarbonyl-Phe-Arg-4-methylcoumaryl-7-amide | - |
Homo sapiens | |
0.05 | - |
Arg-4-methylcoumaryl-7-amide | - |
Homo sapiens | |
0.055 | - |
benzyloxycarbonyl-Arg-Arg-4-methoxy-beta-naphthylamide | - |
Homo sapiens |
Natural Substrates | Organism | Comment (Nat. Sub.) | Natural Products | Comment (Nat. Pro.) | Rev. | Reac. |
---|---|---|---|---|---|---|
Proteins + H2O | Homo sapiens | plays a role in cancer invasion and metastasis | ? | - |
? |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Homo sapiens | - |
- |
- |
Source Tissue | Comment | Organism | Textmining |
---|---|---|---|
breast cancer cell | - |
Homo sapiens | - |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
Arg-4-methylcoumaryl-7-amide + H2O | - |
Homo sapiens | Arg + 7-amino-4-methylcoumarin | - |
? | |
benzyloxycarbonyl-Ala-Arg-Arg-4-methoxy-beta-naphthylamide + H2O | - |
Homo sapiens | benzyloxycarbonyl-Ala-Arg-Arg + 4-methoxy-beta-naphthylamine | - |
? | |
benzyloxycarbonyl-Arg-Arg-4-methoxy-beta-naphthylamide + H2O | - |
Homo sapiens | benzyloxycarbonyl-Arg-Arg + 4-methoxy-beta-naphthylamine | - |
? | |
benzyloxycarbonyl-Arg-Arg-4-methylcoumarin 7-amide + H2O | - |
Homo sapiens | benzyloxycarbonyl-Arg-Arg + 7-amino-4-methylcoumarin | - |
? | |
benzyloxycarbonyl-Arg-Arg-beta-naphthylamide + H2O | - |
Homo sapiens | benzyloxycarbonyl-Arg-Arg + beta-naphthylamine | - |
? | |
benzyloxycarbonyl-Phe-Arg-4-methylcoumarin-7-amide | - |
Homo sapiens | benzyloxycarbonyl-Phe-Arg + 7-amino-4-methylcoumarin | - |
? | |
benzyloxycarbonyl-Val-Lys-Lys-Arg-4-methoxy-beta-naphthylamide + H2O | - |
Homo sapiens | ? + 4-methoxy-beta-naphthylamine | - |
? | |
Collagen + H2O | - |
Homo sapiens | Hydrolyzed collagen | - |
? | |
Proteins + H2O | plays a role in cancer invasion and metastasis | Homo sapiens | ? | - |
? | |
proteoglycans + H2O | - |
Homo sapiens | hydrolyzed proteoglycans | - |
? |
Turnover Number Minimum [1/s] | Turnover Number Maximum [1/s] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|
0.004 | - |
Arg-4-methylcoumaryl-7-amide | - |
Homo sapiens | |
0.125 | - |
benzyloxycarbonyl-Ala-Arg-Arg-4-methoxy-beta-naphthylamide | - |
Homo sapiens | |
0.139 | - |
benzyloxycarbonyl-Arg-Arg-4-methoxy-beta-naphthylamide | - |
Homo sapiens | |
0.149 | - |
benzyloxycarbonyl-Arg-Arg-4-methylcoumaryl-7-amide | - |
Homo sapiens | |
0.325 | - |
benzyloxycarbonyl-Val-Lys-Lys-Arg-4-methoxy-beta-naphthylamide | - |
Homo sapiens | |
0.445 | - |
benzyloxycarbonyl-Phe-Arg-4-methylcoumaryl-7-amide | - |
Homo sapiens |
pH Optimum Minimum | pH Optimum Maximum | Comment | Organism |
---|---|---|---|
6 | - |
- |
Homo sapiens |