Literature summary for 3.4.22.56 extracted from

Guo, Z.; Xian, M.; Zhang, W.; McGill, A.; Wang, P.G.
N-nitrosoanilines: a new class of caspase-3 inhibitors (2001), Bioorg. Med. Chem., 9, 99-106.

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Inhibitors

Inhibitors	Comment	Organism	Structure
m-(Ac-L-Asp-L-Val-NH)-N-nitroso-N-phenylglycine	-	Homo sapiens
N-acetyl-L-alpha-aspartyl-L-valyl-N-[(1S)-2-carboxy-1-[[(4-methylphenyl)(nitroso)amino]methyl]ethyl]-L-alaninamide	-	Homo sapiens
NO	-	Homo sapiens

Organism

Organism	UniProt	Comment	Textmining
Homo sapiens	-	-	-

Substrates and Products (Substrate)

Substrates	Comment Substrates	Organism	Products	Comment (Products)	Rev.	Reac.
acetyl-VDQMDGW-amide + H2O	preferred peptide substrate	Homo sapiens	?	-	?

Ki Value [mM]

Ki Value [mM]	Ki Value maximum [mM]	Inhibitor	Comment	Organism	Structure
0.002	-	N-acetyl-L-alpha-aspartyl-L-valyl-N-[(1S)-2-carboxy-1-[[(4-methylphenyl)(nitroso)amino]methyl]ethyl]-L-alaninamide	pH 7.5, 30°C	Homo sapiens
0.022	-	m-(Ac-L-Asp-L-Val-NH)-N-nitroso-N-phenylglycine	pH 7.5, 37°C	Homo sapiens

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Release 2023.1 (January 2023)