Inhibitors | Comment | Organism | Structure |
---|---|---|---|
(R)-3-(N-benzyloxycarbonylamino)-2-oxo-butylphosphate | - |
Enterobacter cloacae | |
(R)-3-(N-benzyloxycarbonylamino)-2-oxo-butylphosphate | - |
Escherichia coli | |
(RS)-4-(N-benzyloxycarbonyl)amino-3-oxo-2-butylphosphate | - |
Enterobacter cloacae | |
(RS)-4-(N-benzyloxycarbonyl)amino-3-oxo-2-butylphosphate | - |
Escherichia coli | |
3-(N-benzyloxycarbonyl)amino-2-oxopropylphenylphosphonate | - |
Enterobacter cloacae | |
3-(N-benzyloxycarbonyl)amino-2-oxopropylphenylphosphonate | - |
Escherichia coli | |
3-(N-benzyloxycarbonyl)amino-2-oxopropylphosphate | - |
Enterobacter cloacae | |
3-(N-benzyloxycarbonyl)amino-2-oxopropylphosphate | - |
Escherichia coli | |
3-(N-benzyloxycarbonyl)amino-2-oxopropylphosphonate | - |
Enterobacter cloacae | |
3-(N-benzyloxycarbonyl)amino-2-oxopropylphosphonate | - |
Escherichia coli | |
4-(N-benzyloxycarbonyl)amino-3-oxobutylphosphonate | - |
Enterobacter cloacae | |
4-(N-benzyloxycarbonyl)amino-3-oxobutylphosphonate | - |
Escherichia coli | |
ethyl 3-(benzyloxycarbonyl)amino-2-oxo-1,1-difluoropropylphosphonate | - |
Enterobacter cloacae | |
ethyl 3-(benzyloxycarbonyl)amino-2-oxo-1,1-difluoropropylphosphonate | - |
Escherichia coli | |
methyl 3-(N-benzyloxycarbonyl)amino-2-oxo-1-propylphosphate | - |
Enterobacter cloacae | |
methyl 3-(N-benzyloxycarbonyl)amino-2-oxo-1-propylphosphate | - |
Escherichia coli | |
N-[N'-(benzyloxycarbonyl)aminoacetyl]amino-methylphosphonate | - |
Enterobacter cloacae | |
N-[N'-(benzyloxycarbonyl)aminoacetyl]amino-methylphosphonate | - |
Escherichia coli | |
phenyl 3-(N-benzyloxycarbonyl)amino-2-oxopropylphosphate | - |
Enterobacter cloacae | |
phenyl 3-(N-benzyloxycarbonyl)amino-2-oxopropylphosphate | - |
Escherichia coli | |
phenyl 3-(N-benzyloxycarbonyl)amino-2-oxopropylphosphonate | - |
Enterobacter cloacae | |
phenyl 3-(N-benzyloxycarbonyl)amino-2-oxopropylphosphonate | - |
Escherichia coli |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Enterobacter cloacae | - |
- |
- |
Enterobacter cloacae P99 | - |
- |
- |
Escherichia coli | - |
- |
- |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
7beta-aminocephalosporanic acid + H2O | - |
Enterobacter cloacae | (2R)-5-[(acetyloxy)methyl]-2-[(R)-amino(carboxy)methyl]-3,6-dihydro-2H-1,3-thiazine-4-carboxylic acid | - |
? | |
7beta-aminocephalosporanic acid + H2O | - |
Enterobacter cloacae P99 | (2R)-5-[(acetyloxy)methyl]-2-[(R)-amino(carboxy)methyl]-3,6-dihydro-2H-1,3-thiazine-4-carboxylic acid | - |
? | |
7beta-[(thien-2-yl)acetamido]-3-[(4-nitro-3-carboxyphenylthio)methyl]-3-cephem-4-carboxylic acid + H2O | - |
Escherichia coli | (2R)-2-[(R)-carboxy{(E)-[1-hydroxy-2-(thiophen-2-yl)ethylidene]amino}methyl]-5-{[(3-carboxy-4-nitrophenyl)sulfanyl]methyl}-3,6-dihydro-2H-1,3-thiazine-4-carboxylic acid | - |
? |
Synonyms | Comment | Organism |
---|---|---|
beta-lactamase OXA-1 | - |
Escherichia coli |
beta-lactamase OXA-10 | - |
Escherichia coli |
beta-lactamase P99 | - |
Enterobacter cloacae |
Ki Value [mM] | Ki Value maximum [mM] | Inhibitor | Comment | Organism | Structure |
---|---|---|---|---|---|
0.077 | - |
phenyl 3-(N-benzyloxycarbonyl)amino-2-oxopropylphosphonate | - |
Escherichia coli | |
0.088 | - |
(RS)-4-(N-benzyloxycarbonyl)amino-3-oxo-2-butylphosphate | - |
Escherichia coli | |
0.1 | - |
3-(N-benzyloxycarbonyl)amino-2-oxopropylphosphate | - |
Escherichia coli | |
0.11 | - |
phenyl 3-(N-benzyloxycarbonyl)amino-2-oxopropylphosphate | - |
Escherichia coli | |
0.13 | - |
phenyl 3-(N-benzyloxycarbonyl)amino-2-oxopropylphosphonate | - |
Escherichia coli | |
0.13 | - |
phenyl 3-(N-benzyloxycarbonyl)amino-2-oxopropylphosphate | - |
Escherichia coli | |
0.15 | - |
3-(N-benzyloxycarbonyl)amino-2-oxopropylphenylphosphonate | - |
Escherichia coli | |
0.15 | - |
3-(N-benzyloxycarbonyl)amino-2-oxopropylphosphonate | - |
Escherichia coli | |
0.19 | - |
3-(N-benzyloxycarbonyl)amino-2-oxopropylphenylphosphonate | - |
Escherichia coli | |
0.2 | - |
(RS)-4-(N-benzyloxycarbonyl)amino-3-oxo-2-butylphosphate | - |
Escherichia coli | |
0.24 | - |
methyl 3-(N-benzyloxycarbonyl)amino-2-oxo-1-propylphosphate | - |
Escherichia coli | |
0.3 | - |
(R)-3-(N-benzyloxycarbonylamino)-2-oxo-butylphosphate | - |
Escherichia coli | |
0.36 | - |
(R)-3-(N-benzyloxycarbonylamino)-2-oxo-butylphosphate | - |
Escherichia coli | |
0.43 | - |
N-[N'-(benzyloxycarbonyl)aminoacetyl]amino-methylphosphonate | - |
Escherichia coli | |
0.47 | - |
4-(N-benzyloxycarbonyl)amino-3-oxobutylphosphonate | - |
Escherichia coli | |
0.6 | - |
3-(N-benzyloxycarbonyl)amino-2-oxopropylphosphate | - |
Escherichia coli | |
0.6 | - |
4-(N-benzyloxycarbonyl)amino-3-oxobutylphosphonate | - |
Escherichia coli | |
0.7 | - |
phenyl 3-(N-benzyloxycarbonyl)amino-2-oxopropylphosphate | - |
Enterobacter cloacae | |
0.73 | - |
3-(N-benzyloxycarbonyl)amino-2-oxopropylphosphonate | - |
Enterobacter cloacae | |
0.93 | - |
ethyl 3-(benzyloxycarbonyl)amino-2-oxo-1,1-difluoropropylphosphonate | - |
Escherichia coli | |
0.93 | - |
N-[N'-(benzyloxycarbonyl)aminoacetyl]amino-methylphosphonate | - |
Enterobacter cloacae | |
0.95 | - |
ethyl 3-(benzyloxycarbonyl)amino-2-oxo-1,1-difluoropropylphosphonate | - |
Enterobacter cloacae | |
0.97 | - |
(RS)-4-(N-benzyloxycarbonyl)amino-3-oxo-2-butylphosphate | - |
Enterobacter cloacae | |
1.13 | - |
methyl 3-(N-benzyloxycarbonyl)amino-2-oxo-1-propylphosphate | - |
Enterobacter cloacae | |
1.23 | - |
4-(N-benzyloxycarbonyl)amino-3-oxobutylphosphonate | - |
Enterobacter cloacae | |
1.59 | - |
phenyl 3-(N-benzyloxycarbonyl)amino-2-oxopropylphosphonate | - |
Enterobacter cloacae | |
2 | - |
3-(N-benzyloxycarbonyl)amino-2-oxopropylphosphate | - |
Enterobacter cloacae | |
2.1 | - |
(R)-3-(N-benzyloxycarbonylamino)-2-oxo-butylphosphate | - |
Enterobacter cloacae | |
5 | - |
3-(N-benzyloxycarbonyl)amino-2-oxopropylphenylphosphonate | - |
Enterobacter cloacae |