Crystallization (Comment) | Organism |
---|---|
the hCA II-sulthiame complex is crystallized by cocrystallization procedures. High resolution crystal structure of the hCA II-sulthiame adduct | Homo sapiens |
Inhibitors | Comment | Organism | Structure |
---|---|---|---|
sulthiame | isoenzyme hCA I; isoenzyme hCA II; isoenzyme hCA III; isoenzyme hCA IV; isoenzyme hCA IX; isoenzyme hCA VA; isoenzyme hCA VB; isoenzyme hCA VI; isoenzyme hCA VII; isoenzyme hCA XIV | Homo sapiens | |
sulthiame | isoenzyme mCA XIII | Mus musculus |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Homo sapiens | P00915 | - |
- |
Homo sapiens | P00918 | - |
- |
Homo sapiens | P07451 | - |
- |
Homo sapiens | P22748 | - |
- |
Homo sapiens | P23280 | - |
- |
Homo sapiens | P35218 | - |
- |
Homo sapiens | P43166 | - |
- |
Homo sapiens | Q16790 | - |
- |
Homo sapiens | Q9ULX7 | - |
- |
Homo sapiens | Q9Y2D0 | - |
- |
Mus musculus | Q9D6N1 | - |
- |
Synonyms | Comment | Organism |
---|---|---|
hCA I | - |
Homo sapiens |
HCA II | - |
Homo sapiens |
hCA III | - |
Homo sapiens |
hCA IV | - |
Homo sapiens |
hCA IX | - |
Homo sapiens |
hCA VA | - |
Homo sapiens |
hCA VB | - |
Homo sapiens |
hCA VI | - |
Homo sapiens |
hCA VII | - |
Homo sapiens |
hCA XIV | - |
Homo sapiens |
mCA XIII | - |
Mus musculus |
Ki Value [mM] | Ki Value maximum [mM] | Inhibitor | Comment | Organism | Structure |
---|---|---|---|---|---|
0.000006 | - |
sulthiame | isoenzyme hCA VII | Homo sapiens | |
0.000007 | - |
sulthiame | isoenzyme hCA II | Homo sapiens | |
0.000043 | - |
sulthiame | isoenzyme hCA IX | Homo sapiens | |
0.000081 | - |
sulthiame | isoenzyme hCA VA | Homo sapiens | |
0.000091 | - |
sulthiame | isoenzyme hCA VB | Homo sapiens | |
0.000095 | - |
sulthiame | isoenzyme hCA IV | Homo sapiens | |
0.000134 | - |
sulthiame | isoenzyme hCA VI | Homo sapiens | |
0.000374 | - |
sulthiame | isoenzyme hCA I | Homo sapiens | |
0.00145 | - |
sulthiame | isoenzyme mCA XIII | Mus musculus | |
0.00525 | - |
sulthiame | isoenzyme hCA XIV | Homo sapiens | |
0.63 | - |
sulthiame | isoenzyme hCA III | Homo sapiens |