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Literature summary for 4.2.1.1 extracted from

  • Hilvo, M.; Innocenti, A.; Monti, S.M.; De Simone, G.; Supuran, C.T.; Parkkila, S.
    Recent advances in research on the most novel carbonic anhydrases, CA XIII and XV (2008), Curr. Pharm. Des., 14, 672-678.
    View publication on PubMed

Inhibitors

Inhibitors Comment Organism Structure
azetazolamide
-
Homo sapiens
azetazolamide
-
Mus musculus

Organism

Organism UniProt Comment Textmining
Homo sapiens
-
-
-
Mus musculus
-
-
-

Substrates and Products (Substrate)

Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
CO2 + H2O
-
Mus musculus H2CO3
-
r
CO2 + H2O
-
Homo sapiens H2CO3
-
r

Synonyms

Synonyms Comment Organism
CA XIII isozyme Homo sapiens
Ca XV isozyme Mus musculus
carbonic anhydrase
-
Mus musculus
carbonic anhydrase
-
Homo sapiens

Turnover Number [1/s]

Turnover Number Minimum [1/s] Turnover Number Maximum [1/s] Substrate Comment Organism Structure
150000
-
CO2
-
Homo sapiens
470000
-
CO2
-
Mus musculus

Ki Value [mM]

Ki Value [mM] Ki Value maximum [mM] Inhibitor Comment Organism Structure
0.000016
-
azetazolamide
-
Homo sapiens
0.000072
-
azetazolamide
-
Mus musculus