Application | Comment | Organism |
---|---|---|
analysis | use of pharmacophore models for the prediction of binding to P-glycoprotein | Homo sapiens |
Cloned (Comment) | Organism |
---|---|
expression in MDCK cell | Homo sapiens |
Inhibitors | Comment | Organism | Structure |
---|---|---|---|
acitretin | - |
Homo sapiens | |
cholecalciferol | - |
Homo sapiens | |
miconazole | - |
Homo sapiens | |
misoprostol | - |
Homo sapiens | |
nafcillin | - |
Homo sapiens | |
repaglinide | - |
Homo sapiens | |
salmeterol | - |
Homo sapiens | |
telmisartan | - |
Homo sapiens |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Homo sapiens | - |
isoform ABCB1 | - |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
ATP + H2O + acitretin/in | - |
Homo sapiens | ADP + phosphate + acitretin/out | - |
? | |
ATP + H2O + misoprostol/in | - |
Homo sapiens | ADP + phosphate + misoprostol/out | - |
? | |
ATP + H2O + repaglinide/in | - |
Homo sapiens | ADP + phosphate + repaglinide/out | - |
? | |
ATP + H2O + salmeterol/in | - |
Homo sapiens | ADP + phosphate + salmeterol/out | - |
? | |
ATP + H2O + telmisartan/in | - |
Homo sapiens | ADP + phosphate + telmisartan/out | - |
? |