EC Number | Inhibitors | Comment | Organism | Structure |
---|---|---|---|---|
1.14.99.29 | 2,2'-dipyridyl | IC50 0.029 mM | Homo sapiens | |
1.14.99.29 | 4,6-diphenyl-1-hydroxy-pyridine-2-one | IC50 0.0007 mM | Homo sapiens | |
1.14.99.29 | ciclopirox | IC50 0.0006 mM | Homo sapiens | |
1.14.99.29 | Co(C2H3O2)2 | above 0.01 mM | Homo sapiens | |
1.14.99.29 | CuCl2 | above 0.01 mM | Homo sapiens | |
1.14.99.29 | EDTA | IC50 0.0003 mM | Homo sapiens | |
1.14.99.29 | metipirox | IC50 0.0028 mM | Homo sapiens | |
1.14.99.29 | mimosine | IC50 0.0033 mM | Homo sapiens | |
1.14.99.29 | Mn(C2H3O2)2 | above 0.001 mM | Homo sapiens | |
1.14.99.29 | additional information | partial reconstitution of chelator inhibited activity with CuCl2 or Zn(C2H3O2)2 | Homo sapiens | |
1.14.99.29 | Ni(C2H3O2)2 | above 0.001 mM | Homo sapiens | |
1.14.99.29 | Zn(C2H3O2)2 | above 0.01 mM | Homo sapiens |
EC Number | Metals/Ions | Comment | Organism | Structure |
---|---|---|---|---|
1.14.99.29 | Fe2+ | 1.5-fold activation at 0.001 mM | Homo sapiens | |
1.14.99.29 | Fe3+ | 1.5-fold activation at 0.001 mM | Homo sapiens |
EC Number | Organism | UniProt | Comment | Textmining |
---|---|---|---|---|
1.14.99.29 | Homo sapiens | - |
- |
- |
EC Number | Source Tissue | Comment | Organism | Textmining |
---|---|---|---|---|
1.14.99.29 | HeLa-S3 cell | - |
Homo sapiens | - |
EC Number | Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|---|
1.14.99.29 | N'-(4-aminobutyl)lysine + electron donor + O2 | i.e. deoxyhypusine | Homo sapiens | N'-(4-amino-2-hydroxybutyl)lysine + oxidized electron donor + H2O | i.e. hypusine | ? |
EC Number | Temperature Optimum [°C] | Temperature Optimum Maximum [°C] | Comment | Organism |
---|---|---|---|---|
1.14.99.29 | 37 | - |
assay at | Homo sapiens |
EC Number | pH Optimum Minimum | pH Optimum Maximum | Comment | Organism |
---|---|---|---|---|
1.14.99.29 | 7.5 | - |
assay in 50 mM sodium phosphate buffer | Homo sapiens |
EC Number | IC50 Value | IC50 Value Maximum | Comment | Organism | Inhibitor | Structure |
---|---|---|---|---|---|---|
1.14.99.29 | 0.0003 | - |
IC50 0.0003 mM | Homo sapiens | EDTA | |
1.14.99.29 | 0.0006 | - |
IC50 0.0006 mM | Homo sapiens | ciclopirox | |
1.14.99.29 | 0.0007 | - |
IC50 0.0007 mM | Homo sapiens | 4,6-diphenyl-1-hydroxy-pyridine-2-one | |
1.14.99.29 | 0.0028 | - |
IC50 0.0028 mM | Homo sapiens | metipirox | |
1.14.99.29 | 0.0033 | - |
IC50 0.0033 mM | Homo sapiens | mimosine | |
1.14.99.29 | 0.029 | - |
IC50 0.029 mM | Homo sapiens | 2,2'-dipyridyl |