EC Number | Application | Comment | Organism |
---|---|---|---|
7.6.2.2 | analysis | use of pharmacophore models for the prediction of binding to P-glycoprotein | Homo sapiens |
EC Number | Cloned (Comment) | Organism |
---|---|---|
7.6.2.2 | expression in MDCK cell | Homo sapiens |
EC Number | Inhibitors | Comment | Organism | Structure |
---|---|---|---|---|
7.6.2.2 | acitretin | - |
Homo sapiens | |
7.6.2.2 | cholecalciferol | - |
Homo sapiens | |
7.6.2.2 | miconazole | - |
Homo sapiens | |
7.6.2.2 | misoprostol | - |
Homo sapiens | |
7.6.2.2 | nafcillin | - |
Homo sapiens | |
7.6.2.2 | repaglinide | - |
Homo sapiens | |
7.6.2.2 | salmeterol | - |
Homo sapiens | |
7.6.2.2 | telmisartan | - |
Homo sapiens |
EC Number | Organism | UniProt | Comment | Textmining |
---|---|---|---|---|
7.6.2.2 | Homo sapiens | - |
isoform ABCB1 | - |
EC Number | Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|---|
7.6.2.2 | ATP + H2O + acitretin/in | - |
Homo sapiens | ADP + phosphate + acitretin/out | - |
? | |
7.6.2.2 | ATP + H2O + misoprostol/in | - |
Homo sapiens | ADP + phosphate + misoprostol/out | - |
? | |
7.6.2.2 | ATP + H2O + repaglinide/in | - |
Homo sapiens | ADP + phosphate + repaglinide/out | - |
? | |
7.6.2.2 | ATP + H2O + salmeterol/in | - |
Homo sapiens | ADP + phosphate + salmeterol/out | - |
? | |
7.6.2.2 | ATP + H2O + telmisartan/in | - |
Homo sapiens | ADP + phosphate + telmisartan/out | - |
? |