EC Number   |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
|---|
   2.1.1.79 | 0.000011 |
- |
A9145C |
- |
485629 |
| 2.1.1.79 | 0.00013 |
- |
dioctylamine |
competitive inhibitor with respect to phospholipids |
685391 |
| 2.1.1.79 | 0.00022 |
- |
sinefungin |
- |
485629 |
| 2.1.1.79 | 0.00026 |
- |
dioctylamine |
uncompetitive inhibitor with respect to S-adenosyl-L-methionine |
685391 |
| 2.1.1.79 | 0.0005 |
- |
sinefungin |
competitive inhibitor with respect to S-adenosyl-L-methionine |
685391 |
| 2.1.1.79 | 0.001 |
- |
A9145C |
- |
485627 |
| 2.1.1.79 | 0.0011 |
- |
(12aS,12bS)-7-fluoro-2,3,5,12,12a,12b-hexahydro-1H,4H-11-oxa-3a,9b-diazabenzo[a]naphtho[2,1,8-cde]azulene |
inhibits CAFS in a mixed-type fashion with respect to phospholipids |
685391 |
| 2.1.1.79 | 0.0014 |
- |
(12aS,12bS)-7-fluoro-2,3,5,12,12a,12b-hexahydro-1H,4H-11-oxa-3a,9b-diazabenzo[a]naphtho[2,1,8-cde]azulene |
inhibits the CFAS non-competitively with respect to AdoMet |
685391 |
| 2.1.1.79 | 0.004 |
- |
N-octyloctan-1-amine |
37°C, pH 7.4 |
678402 |
| 2.1.1.79 | 0.006 |
- |
5'-S-[2-(decylamino)ethyl]-5'-thioadenosine |
apparent inhibition constant when the phospholipids are the variable substrates. Noncompetitive inhibitor with respect to both substrates |
685391 |
