EC Number |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
---|
2.7.7.60 | 0.00000233 |
- |
cefepime |
pH 7.9, 37°C, recombinant enzyme |
761199 |
2.7.7.60 | 0.000007 |
0.000013 |
(1R,3S)-MMV008138 |
pH 7.4, 37°C |
760263 |
2.7.7.60 | 0.0000759 |
- |
rifampicin |
pH 7.9, 37°C, recombinant enzyme |
761199 |
2.7.7.60 | 0.000169 |
- |
domiphen bromide |
pH 7.9, 37°C, recombinant enzyme |
761199 |
2.7.7.60 | 0.00131 |
- |
tunicamycin |
pH 7.9, 37°C, recombinant enzyme |
761199 |
2.7.7.60 | 0.0015 |
- |
fosmidomycin |
pH 7.9, 37°C, recombinant enzyme |
761199 |
2.7.7.60 | 19.6 |
- |
CTP |
wild type enzyme, pH 6.5, 23°C |
661089 |