EC Number |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
---|
3.5.4.3 | 0.0005 |
- |
6-hydroxy-3,4,6,7-tetrahydroimidazo[4,5-e][1,4]diazepine-5,8-dione |
pH 7.4, 25°C |
667985 |
3.5.4.3 | 0.00188 |
- |
2,6-diaminopurine |
in 25 mM Tris-HCl, 137 mM NaCl, 2.7 mM KCl, at pH 7.4 and 25°C |
711469 |
3.5.4.3 | 0.00196 |
- |
xanthine |
in 25 mM Tris-HCl, 137 mM NaCl, 2.7 mM KCl, at pH 7.4 and 25°C |
711469 |
3.5.4.3 | 0.00201 |
- |
3-benzyl-6-(hydroxymethyl)-3,4,6,7-tetrahydroimidazo[4,5-e][1,4]diazepine-5,8-dione |
pH 7.4, 25°C |
667985 |
3.5.4.3 | 0.0025 |
- |
azepinomycin |
at 25°C and pH 7.4 |
733480 |
3.5.4.3 | 0.00344 |
- |
N-2-acetylguanine |
in 25 mM Tris-HCl, 137 mM NaCl, 2.7 mM KCl, at pH 7.4 and 25°C |
711469 |
3.5.4.3 | 0.00434 |
- |
uric acid |
in 25 mM Tris-HCl, 137 mM NaCl, 2.7 mM KCl, at pH 7.4 and 25°C |
711469 |
3.5.4.3 | 0.00444 |
- |
5-amino-4-imidazole carboxamide |
in 25 mM Tris-HCl, 137 mM NaCl, 2.7 mM KCl, at pH 7.4 and 25°C |
711469 |
3.5.4.3 | 0.00536 |
- |
6-(hydroxymethyl)-3,4,6,7-tetrahydroimidazo[4,5-e][1,4]diazepine-5,8-dione |
pH 7.4, 25°C |
667985 |
3.5.4.3 | 0.00555 |
- |
7-methylguanine |
in 25 mM Tris-HCl, 137 mM NaCl, 2.7 mM KCl, at pH 7.4 and 25°C |
711469 |