EC Number |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
---|
1.14.11.29 | 0.0026 |
- |
(2R)-[2-[2-(5-cyano-3-hydroxypyridin-2-yl)-1,3-thiazol-4-yl]acetamido](phenyl)acetic acid |
pH and temperature not specified in the publication |
742072 |
1.14.11.29 | 0.0028 |
- |
(2S)-[2-[2-(5-cyano-3-hydroxypyridin-2-yl)-1,3-thiazol-4-yl]acetamido](phenyl)acetic acid |
pH and temperature not specified in the publication |
742072 |
1.14.11.29 | 0.0295 |
- |
1,1',1'',1'''-(1,4,7,10-tetraazacyclododecane-1,4,7,10-tetrayl)tetrapropan-2-ol |
recombinant enzyme, pH 7.0, 37°C |
725644 |
1.14.11.29 | 0.0397 |
- |
1,1',1'',1'''-(1,4,7,10-tetraazacyclododecane-1,4,7,10-tetrayl)tetrapropan-2-ol |
recombinant enzyme, pH 7.0, 37°C |
726084 |
1.14.11.29 | 0.0309 |
- |
2,2',2'',2'''-(1,4,7,10-tetraazacyclododecane-1,4,7,10-tetrayl)tetraacetamide |
recombinant enzyme, pH 7.0, 37°C |
726084 |
1.14.11.29 | 0.005 |
- |
2,3-dihydroxypyridine |
pH 7.0, 37°C |
725647 |
1.14.11.29 | 0.0004 |
- |
2-(2-(5-cyano-3-hydroxy-4-methylpyridin-2-yl)-5-methylthiazol-4-yl)-N-(2-(diethylamino)ethyl)acetamide |
pH and temperature not specified in the publication |
742072 |
1.14.11.29 | 0.0057 |
- |
2-(2-(5-cyano-3-hydroxy-4-methylpyridin-2-yl)-5-phenylthiazol-4-yl)-N-(2-(pyridin-2-yl)ethyl)acetamide |
pH and temperature not specified in the publication |
742072 |
1.14.11.29 | 0.024 |
- |
2-(2-(5-cyano-3-hydroxypyridin-2-yl)-5-phenylthiazol-4-yl)-N-(2-(pyridin-2-yl)ethyl)acetamide |
pH and temperature not specified in the publication |
742072 |
1.14.11.29 | 0.003 |
- |
2-hydroxypyridine 1-oxide |
pH 7.0, 37°C |
725647 |