EC Number |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
---|
1.1.1.145 | 0.00019 |
- |
(+)-gossypol |
in PBS buffer, pH 7.2 |
699845 |
1.1.1.145 | 0.0002 |
- |
epostane |
in 0.02 M potassium phosphate buffer, pH 7.4 |
700182 |
1.1.1.145 | 0.00023 |
- |
(-)-gossypol |
in PBS buffer, pH 7.2 |
699845 |
1.1.1.145 | 0.0005 |
- |
(1R,9aR,11aR)-9a,11a-dimethyl-1-((R)-6-methylheptan-2-yl)-3,3a,3b,4,5,8,9,9a,9b,10,11,11a-dodecahydro-1H-cyclopenta[i]phenanthridin-7(2H)-one |
pH 8.5, 30°C |
724518 |
1.1.1.145 | 0.0008 |
- |
(1R,4S,9aR,11aR)-4,9a,11a-trimethyl-1-((R)-6-methylheptan-2-yl)-3,3a,3b,4,5,8,9,9a,9b,10,11,11a-dodecahydro-1H-cyclopenta[i]phenanthridin-7(2H)-one |
pH 8.5, 30°C |
724518 |
1.1.1.145 | 0.0027 |
- |
quercetin |
pH 7.4, 25°C |
684725 |
1.1.1.145 | 0.00277 |
- |
(-)-gossypol |
in PBS buffer, pH 7.2 |
699845 |
1.1.1.145 | 0.00445 |
- |
(+)-gossypol |
in PBS buffer, pH 7.2 |
699845 |
1.1.1.145 | 0.0049 |
- |
trilostane |
in 0.02 M potassium phosphate buffer, pH 7.4 |
700182 |
1.1.1.145 | 0.0059 |
- |
genistein |
pH 7.4, 25°C |
684725 |