EC Number |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
---|
3.4.19.12 | 0.00074 |
- |
ubiquitin |
- |
677540 |
3.4.19.12 | 0.00081 |
- |
(3E)-5-bromo-1-(3,4-dichlorobenzyl)-1H-indole-2,3-dione 3-(O-acetyloxime) |
IC50: 0.00081 mM |
664573 |
3.4.19.12 | 0.00088 |
- |
(3E)-5-chloro-1-(2,5-dichlorobenzyl)-1H-indole-2,3-dione 3-(O-acetyloxime) |
IC50: 0.00088 mM |
664573 |
3.4.19.12 | 0.00094 |
- |
(3E)-1-(3,4-dichlorobenzyl)-5-iodo-1H-indole-2,3-dione 3-(O-acetyloxime) |
IC50: 0.00094 mM |
664573 |
3.4.19.12 | 0.0012 |
- |
(3E)-5-chloro-1-(2,4-dichlorobenzyl)-1H-indole-2,3-dione 3-(O-acetyloxime) |
IC50: 0.0012 mM |
664573 |
3.4.19.12 | 0.0013 |
- |
(3E)-5-chloro-1-(3,5-dichlorobenzyl)-1H-indole-2,3-dione 3-(O-acetyloxime) |
IC50: 0.0013 mM |
664573 |
3.4.19.12 | 0.0013 |
- |
(3E)-5-chloro-1-[2-(3,4-dichlorophenyl)ethyl]-1H-indole-2,3-dione 3-(O-acetyloxime) |
IC50: 0.0013 mM |
664573 |
3.4.19.12 | 0.0018 |
- |
(3E)-5-chloro-1-(3,4-dichlorobenzyl)-1H-indole-2,3-dione 3-(O-acetyloxime) |
IC50: 0.0018 mM |
664573 |
3.4.19.12 | 0.0018 |
- |
5-chloro-1-(3,4-dichlorobenzyl)-1H-indole-2,3-dione 3-(O-acetyloxime) |
IC50: 0.0018 mM |
664573 |
3.4.19.12 | 0.0027 |
- |
(3E)-5-chloro-1-(2,3-dichlorobenzyl)-1H-indole-2,3-dione 3-(O-acetyloxime) |
IC50: 0.0027 mM |
664573 |