Inhibitors | Comment | Organism | Structure |
---|---|---|---|
adaptaquin | EC50 of ca 2 mM in HIF1 ODD-luc fusion reporter assay | Homo sapiens | |
N-[(3,4-dimethoxyphenyl)(8-hydroxyquinolin-7-yl)methyl]-2-phenylacetamide | optimized adaptaquin analog, shows no toxicity up to a 100fold increased range over EC50. The drug is ismetabolized by CYP3A4 and CYP2B6 | Homo sapiens |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Homo sapiens | - |
- |
- |
Source Tissue | Comment | Organism | Textmining |
---|---|---|---|
Hepa-RG cell | - |
Homo sapiens | - |