Crystallization (Comment) | Organism |
---|---|
CoMFA and quantum chemical calculations studies on pyrimethamine derivatives active against quadruple mutant N5I/C59R/S108N/I164L. Residue N108 is the cause of pyrimethamine resistance with the highest repulsive interaction energy | Plasmodium falciparum |
Protein Variants | Comment | Organism |
---|---|---|
N5I/C59R/S108N/I164L | naturally occuring mutant. Residue N108 is the cause of pyrimethamine resistance with the highest repulsive interaction energy | Plasmodium falciparum |
Inhibitors | Comment | Organism | Structure |
---|---|---|---|
pyrimethamine | CoMFA and quantum chemical calculations studies on pyrimethamine derivatives active against quadruple mutant N5I/C59R/S108N/I164L. Residue N108 is the cause of pyrimethamine resistance with the highest repusive interaction energy | Plasmodium falciparum |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Plasmodium falciparum | P13922 | - |
- |