Activating Compound | Comment | Organism | Structure |
---|---|---|---|
Diazoacetylnorleucine methyl ester | 1.0 mM, activation to 115% of control | Alitta virens | |
diisopropylphosphoryl fluoride | 1.0 mM, activation to 116.3% of control | Alitta virens | |
Soybean trypsin inhibitor | 0.5 mM, activation to 115% of control | Alitta virens | |
tosylphenylalanine chloromethyl ketone | 1.0 mM, activation to 113% of control | Alitta virens |
Inhibitors | Comment | Organism | Structure |
---|---|---|---|
1,10-phenanthroline | 5.0 mM, complete inhibition | Alitta virens | |
antipain | 0.1 mg/ml, 26% inhibition | Alitta virens | |
captopril | 0.1 mM, complete inhibition | Alitta virens | |
CuCl2 | 73% inhibition at 0.1 mM, 99% inhibition at 1.0 mM | Alitta virens | |
EDTA | 1.0 mM, complete inhibition | Alitta virens | |
leupeptin | 0.1 mg/ml, 18% inhibition | Alitta virens | |
lisinopril | - |
Alitta virens | |
additional information | enzyme is not affected by addition of 0.1-1.0 mM CaCl2, Mn2Cl2, MgCl2 or 0.1 mM ZnCl2 | Alitta virens | |
PCMB | 1.0 mM, 42% inhibition | Alitta virens | |
ZnCl2 | 1.0 mM, 98% inhibition | Alitta virens |
KM Value [mM] | KM Value Maximum [mM] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|
0.56 | - |
benzoyl-Gly-His-Leu | - |
Alitta virens |
Metals/Ions | Comment | Organism | Structure |
---|---|---|---|
CoCl2 | 0.1-1.0 mM, 2fold activation | Alitta virens | |
additional information | enzyme is not affected by addition of 0.1-1.0 mM CaCl2, Mn2Cl2, MgCl2 or 0.1 mM ZnCl2 | Alitta virens |
Molecular Weight [Da] | Molecular Weight Maximum [Da] | Comment | Organism |
---|---|---|---|
69000 | - |
gel filtration | Alitta virens |
71000 | - |
1 * 71000, SDS-PAGE | Alitta virens |
Natural Substrates | Organism | Comment (Nat. Sub.) | Natural Products | Comment (Nat. Pro.) | Rev. | Reac. |
---|---|---|---|---|---|---|
angiotensin I + H2O | Alitta virens | the enzyme plays an important role in blood pressure homeostasis | angiotensin II + His-Leu | - |
? |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Alitta virens | - |
- |
- |
Purification (Comment) | Organism |
---|---|
- |
Alitta virens |
Specific Activity Minimum [µmol/min/mg] | Specific Activity Maximum [µmol/min/mg] | Comment | Organism |
---|---|---|---|
466.8 | - |
- |
Alitta virens |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
angiotensin I + H2O | - |
Alitta virens | angiotensin II + His-Leu | - |
? | |
angiotensin I + H2O | the enzyme plays an important role in blood pressure homeostasis | Alitta virens | angiotensin II + His-Leu | - |
? | |
Arg-Pro-Lys-Pro-Gln-Gln-Phe-Phe-Gly-Leu-Met-NH2 + H2O | cleavage sites: Arg-Pro-/-Lys-Pro-/-Gln-Gln-/-Phe-Phe-/-Gly-Leu-Met-NH2 | Alitta virens | ? | - |
? | |
bradykinin + H2O | - |
Alitta virens | Phe-Arg + Ser-Pro + Arg-Pro-Pro-Gly-Phe | - |
? | |
hippuryl-Gly-His-Leu + H2O | - |
Alitta virens | hippuric acid + His-Leu | - |
? | |
hippuryl-His-Leu + H2O | - |
Alitta virens | hippuric acid + His-Leu | - |
? | |
additional information | no cleavage of imido-bonds. No hydrolysis of angiotensin II and angiotensin III | Alitta virens | ? | - |
? | |
Tyr-Gly-Gly-Phe-Leu + H2O | - |
Alitta virens | Tyr-Gly-Gly + Phe-Leu | - |
? | |
Tyr-Gly-Gly-Phe-Met + H2O | - |
Alitta virens | Tyr-Gly-Gly + Phe-Met | - |
? |
Subunits | Comment | Organism |
---|---|---|
monomer | 1 * 71000, SDS-PAGE | Alitta virens |
Synonyms | Comment | Organism |
---|---|---|
DCP | - |
Alitta virens |
Temperature Optimum [°C] | Temperature Optimum Maximum [°C] | Comment | Organism |
---|---|---|---|
45 | - |
- |
Alitta virens |
Turnover Number Minimum [1/s] | Turnover Number Maximum [1/s] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|
345 | - |
benzoyl-Gly-His-Leu | - |
Alitta virens |
pH Optimum Minimum | pH Optimum Maximum | Comment | Organism |
---|---|---|---|
8 | - |
- |
Alitta virens |
Ki Value [mM] | Ki Value maximum [mM] | Inhibitor | Comment | Organism | Structure |
---|---|---|---|---|---|
0.00000138 | - |
captopril | - |
Alitta virens | |
0.00000207 | - |
lisinopril | - |
Alitta virens |
Organism | Comment | pI Value Maximum | pI Value |
---|---|---|---|
Alitta virens | - |
- |
4.5 |