Activating Compound | Comment | Organism | Structure |
---|---|---|---|
ubiquitin | submicromolar concentrations activate while higher concentrations inhibit the enzyme, regulatory function, binding via 2 ubiquitin binding sites extending the active site | Oryctolagus cuniculus |
Inhibitors | Comment | Organism | Structure |
---|---|---|---|
ubiquitin | submicromolar concentrations activate while higher concentrations inhibit the enzyme, regulatory function, 2-step inhibition mechanism via 2 ubiquitin binding sites extending the active site | Oryctolagus cuniculus | |
Ubiquitin aldehyde | inhibition in absence of ubiquitin, competitive to ubiquitin | Oryctolagus cuniculus |
KM Value [mM] | KM Value Maximum [mM] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|
additional information | - |
additional information | kinetics | Oryctolagus cuniculus |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Oryctolagus cuniculus | - |
- |
- |
Source Tissue | Comment | Organism | Textmining |
---|---|---|---|
reticulocyte | - |
Oryctolagus cuniculus | - |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
polyubiquitin + H2O | - |
Oryctolagus cuniculus | ubiquitin | - |
? |
Temperature Optimum [°C] | Temperature Optimum Maximum [°C] | Comment | Organism |
---|---|---|---|
25 | - |
assay at | Oryctolagus cuniculus |
pH Optimum Minimum | pH Optimum Maximum | Comment | Organism |
---|---|---|---|
7.8 | - |
assay at | Oryctolagus cuniculus |
Ki Value [mM] | Ki Value maximum [mM] | Inhibitor | Comment | Organism | Structure |
---|---|---|---|---|---|
additional information | - |
additional information | inhibition kinetics | Oryctolagus cuniculus | |
0.0000001 | - |
ubiquitin-aldehyde | at 0.0006 mM ubiquitin, pH 7.8, 25°C | Oryctolagus cuniculus | |
0.0000023 | - |
ubiquitin-aldehyde | in absence of ubiquitin, pH 7.8, 25°C | Oryctolagus cuniculus |