EC Number |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
---|
1.13.11.27 | 0.0013 |
- |
(2,6-difluoro-4-hydroxyphenyl)pyruvate |
- |
395372 |
1.13.11.27 | 0.000102 |
- |
(3-cyclopropyl-5-hydroxy-1-methyl-1H-pyrazol-4-yl)(5,7-dichlorobenzofuran-2-yl)methanone |
30°C, pH not specified in the publication |
765504 |
1.13.11.27 | 0.000099 |
- |
(3-cyclopropyl-5-hydroxy-1-methyl-1H-pyrazol-4-yl)(5-nitrobenzofuran-2-yl)methanone |
30°C, pH not specified in the publication |
765504 |
1.13.11.27 | 0.000223 |
- |
(5,7-dichlorobenzofuran-2-yl)(5-hydroxy-1-methyl-3-(trifluoromethyl)-1H-pyrazol-4-yl)methanone |
30°C, pH not specified in the publication |
765504 |
1.13.11.27 | 0.000458 |
- |
1-benzyl-6-(2-hydroxy-4,4-dimethyl-6-oxocyclohex-1-ene-1-carbonyl)-3-(4-methylphenyl)quinazoline-2,4(1H,3H)-dione |
recombinant His-tagged enzyme, pH 7.0, 30°C |
743407 |
1.13.11.27 | 0.000355 |
- |
1-benzyl-6-(2-hydroxy-6-oxocyclohex-1-ene-1-carbonyl)-3-(4-methylphenyl)quinazoline-2,4(1H,3H)-dione |
recombinant His-tagged enzyme, pH 7.0, 30°C |
743407 |
1.13.11.27 | 0.000028 |
- |
1-butyl-6-(2-hydroxy-4,4-dimethyl-6-oxocyclohex-1-ene-1-carbonyl)-3-(4-methylphenyl)quinazoline-2,4(1H,3H)-dione |
recombinant His-tagged enzyme, pH 7.0, 30°C |
743407 |
1.13.11.27 | 0.000019 |
- |
1-butyl-6-(2-hydroxy-6-oxocyclohex-1-ene-1-carbonyl)-3-(4-methylphenyl)quinazoline-2,4(1H,3H)-dione |
recombinant His-tagged enzyme, pH 7.0, 30°C |
743407 |
1.13.11.27 | 0.000045 |
- |
1-ethyl-6-(2-hydroxy-4,4-dimethyl-6-oxocyclohex-1-ene-1-carbonyl)-3-(4-methylphenyl)quinazoline-2,4(1H,3H)-dione |
recombinant His-tagged enzyme, pH 7.0, 30°C |
743407 |
1.13.11.27 | 0.000047 |
- |
1-ethyl-6-(2-hydroxy-4-methyl-6-oxocyclohex-1-ene-1-carbonyl)-3-(4-methylphenyl)quinazoline-2,4(1H,3H)-dione |
recombinant His-tagged enzyme, pH 7.0, 30°C |
743407 |