EC Number |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
---|
3.4.24.17 | 0.00000013 |
- |
tissue inhibitor of metalloproteinases 1 |
catalytic enzyme domain, pH 7.0, 37°C |
734175 |
3.4.24.17 | 0.00000055 |
- |
tissue inhibitor of metalloproteinases 2 |
catalytic enzyme domain, pH 7.0, 37°C |
734175 |
3.4.24.17 | 0.000002 |
- |
2-Butyl-4-[2,2-dimethyl-1-(pyridin-4-ylcarbamoyl)-propylcarbamoyl]-6-(4'-fluoro-biphenyl-4-yl)-hexanoic acid |
pH 6.5, 25°C |
652709 |
3.4.24.17 | 0.000004 |
- |
2-Butyl-4-(2,2-dimethyl-1-phenylcarbamoyl-propylcarbamoyl)-6-(4'-fluoro-biphenyl-4-yl)-hexanoic acid |
pH 6.5, 25°C |
652709 |
3.4.24.17 | 0.000005 |
- |
2-Butyl-4-[(2,2-dimethyl-1-methylcarbamoyl-propylamino)-hydroxy-methyl]-6-(4'-methylsulfanyl-biphenyl-4-yl)-hexanoic acid |
pH 6.5, 25°C |
652709 |
3.4.24.17 | 0.000009 |
- |
2-Butyl-6-(4'-cyano-biphenyl-4-yl)-4-[(2,2-dimethyl-1-methylcarbamoyl-propylamino)-hydroxy-methyl]-hexanoic acid |
pH 6.5, 25°C |
652709 |
3.4.24.17 | 0.00001 |
- |
2-Butyl-4-(2,2-dimethyl-1-methylcarbamoyl-propylcarbamoyl)-6-(4'-fluoro-biphenyl-4-yl)-hexanoic acid |
pH 6.5, 25°C |
652709 |
3.4.24.17 | 0.000011 |
- |
2-Butyl-4-[(2,2-dimethyl-1-methylcarbamoyl-propylamino)-hydroxy-methyl]-6-(2'-fluoro-biphenyl-4-yl)-hexanoic acid |
pH 6.5, 25°C |
652709 |
3.4.24.17 | 0.000011 |
- |
2-Butyl-4-[2,2-dimethyl-1-(pyridin-4-ylcarbamoyl)-propylcarbamoyl]-6-(4-propyl-phenyl)-hexanoic acid |
pH 6.5, 25°C |
652709 |
3.4.24.17 | 0.000011 |
- |
6-(4'-Bromo-biphenyl-4-yl)-2-butyl-4-[(2,2-dimethyl-1-methylcarbamoyl-propylamino)-hydroxy-methyl]-hexanoic acid |
pH 6.5, 25°C |
652709 |