EC Number   |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference  |
|---|
   1.14.11.29 | 0.04 |
- |
3-hydroxy-1,2-dimethyl-4(1H)-pyridinone |
pH 7.0, 37°C |
725647 |
| 1.14.11.29 | 0.4 |
- |
5-hydroxy-2-hydroxymethyl-4-pyrone |
pH 7.0, 37°C |
725647 |
| 1.14.11.29 | 1 |
- |
3-cyano-6-methyl-2(H)-pyridinone |
above, pH 7.0, 37°C |
725647 |
| 1.14.11.29 | 1 |
- |
3-hydroxy-2-methyl-4-pyrone |
above, pH 7.0, 37°C |
725647 |
| 1.14.11.29 | 0.0103 |
- |
3,6,9-tris(naphthalen-1-ylmethyl)-3,6,9,15-tetraazabicyclo[9.3.1]pentadeca-1(15),11,13-triene |
recombinant enzyme, pH 7.0, 37°C |
726084 |
| 1.14.11.29 | 0.0207 |
- |
N,N-dimethyl-5-[3,6,9,15-tetraazabicyclo[9.3.1]pentadeca-1(15),11,13-trien-6-ylsulfonyl]naphthalen-1-amine |
recombinant enzyme, pH 7.0, 37°C |
726084 |
| 1.14.11.29 | 0.0309 |
- |
2,2',2'',2'''-(1,4,7,10-tetraazacyclododecane-1,4,7,10-tetrayl)tetraacetamide |
recombinant enzyme, pH 7.0, 37°C |
726084 |
| 1.14.11.29 | 0.0397 |
- |
1,1',1'',1'''-(1,4,7,10-tetraazacyclododecane-1,4,7,10-tetrayl)tetrapropan-2-ol |
recombinant enzyme, pH 7.0, 37°C |
726084 |
| 1.14.11.29 | 0.0004 |
- |
2-(2-(5-cyano-3-hydroxy-4-methylpyridin-2-yl)-5-methylthiazol-4-yl)-N-(2-(diethylamino)ethyl)acetamide |
pH and temperature not specified in the publication |
742072 |
| 1.14.11.29 | 0.0007 |
- |
2-[2-(5-cyano-3-hydroxy-4-methylpyridin-2-yl)-1,3-thiazol-4-yl]-N-[2-(pyridin-2-yl)ethyl]acetamide |
pH and temperature not specified in the publication |
742072 |
