EC Number |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
---|
1.7.1.B2 | 0.2 |
- |
5-(aziridin-1-yl)-2,4-dinitrobenzamide |
mutant enzyme T41L/F70A/F108Y, at pH 7.0 and 23°C |
764166 |
1.7.1.B2 | 0.23 |
- |
2-(2-methyl-5-nitro-1H-imidazol-1-yl)-N-(2,2,3,3,3-pentafluoropropyl)acetamide |
mutant enzyme E72Q/F108Y, at pH 7.0 and 23°C |
764166 |
1.7.1.B2 | 0.23 |
- |
5-(aziridin-1-yl)-2,4-dinitrobenzamide |
mutant enzyme T41L/F70A, at pH 7.0 and 23°C |
764166 |
1.7.1.B2 | 0.25 |
- |
5-(aziridin-1-yl)-2,4-dinitrobenzamide |
mutant enzyme T41L/F70A/N71S, at pH 7.0 and 23°C |
764166 |
1.7.1.B2 | 0.26 |
- |
2-(2-methyl-5-nitro-1H-imidazol-1-yl)-N-(2,2,3,3,3-pentafluoropropyl)acetamide |
mutant enzyme F108Y, at pH 7.0 and 23°C |
764166 |
1.7.1.B2 | 0.29 |
- |
5-(aziridin-1-yl)-2,4-dinitrobenzamide |
mutant enzyme T41L, at pH 7.0 and 23°C |
764166 |
1.7.1.B2 | 0.31 |
- |
2-(2-methyl-5-nitro-1H-imidazol-1-yl)-N-(2,2,3,3,3-pentafluoropropyl)acetamide |
mutant enzyme T41L/F70A/N71S, at pH 7.0 and 23°C |
764166 |
1.7.1.B2 | 0.32 |
- |
5-(aziridin-1-yl)-2,4-dinitrobenzamide |
mutant enzyme T41L/F70A/N71S/F108Y, at pH 7.0 and 23°C |
764166 |
1.7.1.B2 | 0.33 |
- |
2,4-dinitrotoluene |
at pH 8.0 and 30°C |
764364 |
1.7.1.B2 | 0.38 |
- |
5-(aziridin-1-yl)-2,4-dinitrobenzamide |
wild type enzyme, at pH 7.0 and 23°C |
764166 |